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Found 66 with Last Name = 'mcpherson' and Initial = 'dw'
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.120nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.160nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50296314((3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carb...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.230nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.260nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  0.270nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405720(CHEMBL2115342)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50296314((3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carb...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.5nMAssay Description:Evaluated for the phosphatidyl inositol turnover at Muscarinic acetylcholine receptor M1 in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50367742(CHEMBL1788199)
Affinity DataKi:  0.570nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.760nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  0.780nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  2.20nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405717(CHEMBL2115341)
Affinity DataKi:  2.90nMAssay Description:Pseudo hill coefficient at Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  5.20nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50367741(CHEMBL1788286)
Affinity DataKi:  5.20nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50367742(CHEMBL1788199)
Affinity DataKi:  5.80nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405720(CHEMBL2115342)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405720(CHEMBL2115342)
Affinity DataKi:  6.90nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50296314((3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carb...)
Affinity DataKi:  6.90nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  7.5nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405718(CHEMBL2114396)
Affinity DataKi:  19nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50367741(CHEMBL1788286)
Affinity DataKi:  27nMAssay Description:Evaluated for the phosphatidyl inositol turnover at Muscarinic acetylcholine receptor M1 in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405717(CHEMBL2115341)
Affinity DataKi:  37nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50367741(CHEMBL1788286)
Affinity DataKi:  74nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50367742(CHEMBL1788199)
Affinity DataKi:  123nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405720(CHEMBL2115342)
Affinity DataKi:  153nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic receptor M1(Bos taurus)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405719(CHEMBL2114395)
Affinity DataKi:  156nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M1 by displacement of [3H]pirenzepine in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228362(CHEMBL1202960)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228375(CHEMBL1202955)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  267nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  377nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405718(CHEMBL2114396)
Affinity DataKi:  934nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405719(CHEMBL2114395)
Affinity DataKi:  1.37E+3nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor M2 by displacement of [3H]QNB in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50405717(CHEMBL2115341)
Affinity DataKi:  1.46E+3nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228357(CHEMBL1202954)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50367741(CHEMBL1788286)
Affinity DataKi:  1.66E+3nMAssay Description:Evaluated for the inhibition of adenylate cyclase at M2 receptor in rat heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228377(CHEMBL1202958)
Affinity DataKi:  2.38E+3nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228354(CHEMBL557216)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228376(CHEMBL320755)
Affinity DataKi:  5.24E+3nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228355(CHEMBL1202956)
Affinity DataKi:  8.28E+3nMAssay Description:Displacement of [3H]QNB from rat ileum Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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