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Found 187 with Last Name = 'meade' and Initial = 'r'
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298756((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.640nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50035384(Benzyl-[2-(5-bromo-2,3-dimethoxy-phenyl)-3H-imidaz...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]YM-09151 from recombinant African green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048233(1-(2-Methoxy-phenyl)-4-(1-phenyl-1H-pyrrol-3-ylmet...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048240(1-(2-Methoxy-phenyl)-4-(1-methyl-5-phenyl-1H-pyrro...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50048233(1-(2-Methoxy-phenyl)-4-(1-phenyl-1H-pyrrol-3-ylmet...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50048230(1-(1-Phenyl-1H-pyrrol-3-ylmethyl)-4-pyridin-2-yl-p...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM85136(CAS_188942 | CHEMBL103772 | NGD 94-1 | NSC_188942)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298754((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Chlorocebus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-YM 09151 from african moonkey Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298760(CHEMBL574766 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM85136(CAS_188942 | CHEMBL103772 | NGD 94-1 | NSC_188942)
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM85136(CAS_188942 | CHEMBL103772 | NGD 94-1 | NSC_188942)
Affinity DataKi:  3.80nMAssay Description:Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298738(CHEMBL583783 | benzyl(2S,5S,8S,11S,14S)-8-(3-amino...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50048237(4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-1,2,3,6...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50048234(1-Phenyl-4-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperaz...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298761(CHEMBL574788 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]YM-09151 from recombinant African green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity on human Dopamine receptor D2 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50035388(Benzyl-[2-(2,3-dimethoxy-phenyl)-3H-imidazol-4-ylm...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]YM-09151 from recombinant African green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50055810(1-Phenyl-4-(2-phenyl-3H-imidazol-4-ylmethyl)-piper...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298757((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048237(4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-1,2,3,6...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50055807(2-[4-(5-Methyl-2-phenyl-3H-imidazol-4-ylmethyl)-pi...)
Affinity DataKi:  6nMAssay Description:Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298762(CHEMBL574924 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298739(CHEMBL583784 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  7.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50055808(1-(2-Phenyl-3H-imidazol-4-ylmethyl)-4-pyridin-2-yl...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298740(CHEMBL574324 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  8.80nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50048235(4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperid...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Chlorocebus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048233(1-(2-Methoxy-phenyl)-4-(1-phenyl-1H-pyrrol-3-ylmet...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-YM 09151 from african moonkey Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298714(CHEMBL574925 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  11.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298715(CHEMBL575847 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  12.8nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298716(CHEMBL574792 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  13.1nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298741(CHEMBL574931 | benzyl(2S,5S,8S,11S,14S)-7-cyclohex...)
Affinity DataKi:  13.1nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298717(CHEMBL574845 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  13.7nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048234(1-Phenyl-4-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperaz...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Chlorocebus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048237(4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-1,2,3,6...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-YM 09151 from african moonkey Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by PDSP Ki Database
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298742(CHEMBL583785 | benzyl(2S,5S,8S,11S,14S)-8-(2-amino...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298718(CHEMBL574926 | benzyl(2S,5S,8S,11S,14S)-11-((1H-im...)
Affinity DataKi:  18.6nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298755((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  19.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298743(CHEMBL573527 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  19.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Cercopithecus aethiops)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50048235(4-Phenyl-1-(1-phenyl-1H-pyrrol-3-ylmethyl)-piperid...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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