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Found 930 with Last Name = 'meier' and Initial = 'h'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM21244(2-[(1S,2S,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM21244(2-[(1S,2S,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM21244(2-[(1S,2S,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM86515(CAS_1972-08-3 | NSC_16078 | THC, delta 9 | US94161...)
Affinity DataKi:  13.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM86515(CAS_1972-08-3 | NSC_16078 | THC, delta 9 | US94161...)
Affinity DataKi:  22.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  45.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  55.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Bayer Healthcare

Curated by PDSP Ki Database
LigandPNGBDBM86515(CAS_1972-08-3 | NSC_16078 | THC, delta 9 | US94161...)
Affinity DataKi:  69.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Schering

Curated by ChEMBL
LigandPNGBDBM50409115(LONAPRISAN)
Affinity DataIC50:  0.00250nMAssay Description:In vitro antagonist potency in transactivation assay in neuroblastoma cells expressing human PR-B progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Schering

Curated by ChEMBL
LigandPNGBDBM50409115(LONAPRISAN)
Affinity DataIC50:  0.00360nMAssay Description:In vitro antagonist potency in transactivation assay in neuroblastoma cells expressing human PR-A progesterone receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Schering

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.0250nMAssay Description:In vitro antagonist potency in transactivation assay in neuroblastoma cells expressing human PR-B progesterone receptorMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Schering

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataIC50:  0.0280nMAssay Description:In vitro antgonist potency in transactivation assay in neuroblastoma cells expressing human PR-A progesterone receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50327343(2-(4-(8-fluoroquinoxalin-6-yl)-3-methyl-1-o-tolyl-...)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity at adenosine A1 receptor by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255962(US9481672, 140)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255964(US9481672, 142)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine kinase(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50143581(7-[4-(4-Fluoro-benzyl)-[1,4]diazepan-1-yl]-2-pheny...)
Affinity DataIC50: >1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50143575(7-(1-Benzyl-hexahydro-pyrrolo[3,4-b]pyrrol-5-yl)-2...)
Affinity DataIC50: >1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50143574(7-((4aS,7aS)-6-Benzyl-octahydro-pyrrolo[3,4-b]pyri...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256099(US9481672, 281)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256065(US9481672, 247)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256064(US9481672, 246)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255968(US9481672, 146)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256036(US9481672, 217)
Affinity DataIC50:  1nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium channel subfamily K member 9(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM458963((4-{[2-(4-Bromophenyl)imidazo[,2-a]pyridin-3-yl]me...)
Affinity DataIC50:  1.04nMAssay Description:The investigations on the inhibition of the recombinant TASK-1 and TASK-3 channels were carried out using stably transfected CHO cells. Here, the com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Bayer Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50327327(2-(4-(4-fluorophenyl)-3-methyl-1-o-tolyl-1H-pyrazo...)
Affinity DataIC50:  1.39nMAssay Description:Antagonist activity at adenosine A1 receptor by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Bayer

Curated by ChEMBL
LigandPNGBDBM50143592(7-((3aS,6aS)-1-Benzyl-hexahydro-pyrrolo[3,4-b]pyrr...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory activity against human adenosine kinase expressed in E. coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin

Curated by ChEMBL
LigandPNGBDBM50344356(CHEMBL1779676 | ethyl 3-(3-(7-hydroxynaphthalen-1-...)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin

Curated by ChEMBL
LigandPNGBDBM50344356(CHEMBL1779676 | ethyl 3-(3-(7-hydroxynaphthalen-1-...)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM88376(US9695131, 13)
Affinity DataIC50:  1.80nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin

Curated by ChEMBL
LigandPNGBDBM50344367(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-hydrox...)
Affinity DataIC50:  1.90nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255927(US9481672, 104)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255944(US9481672, 122)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256116(US9481672, 300)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256111(US9481672, 294)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256095(US9481672, 277)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256088(BDBM256092 | BDBM256093 | US9481672, 270)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256083(US9481672, 265)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256066(US9481672, 248)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256062(US9481672, 244)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM256059(US9481672, 241)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255954(US9481672, 132)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255956(US9481672, 134)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255958(US9481672, 136)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255961(US9481672, 139)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255963(US9481672, 141)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255965(US9481672, 143)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255966(US9481672, 144)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255967(US9481672, 145)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255969(US9481672, 147)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Targetchymase(Mesocricetus auratus (Golden hamster))
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM255971(US9481672, 149)
Affinity DataIC50:  2nMpH: 7.5Assay Description:The enzyme source used is recombinant human chymase (expressed in HEK293 cells) or chymase purified from hamsters' tongues. The substrate used for ch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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