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Found 75 with Last Name = 'michalewsky' and Initial = 'j'
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003204(CHEMBL122438 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.0290nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003669(Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-Phe-NH2 | CHEMB...)
Affinity DataIC50:  0.0500nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003199(CHEMBL126008 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.0850nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011545(CHEMBL430906 | Desamino-Tyr(SO3H)-Met-Gly-Trp-Met-...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003202(CHEMBL331408 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406497(CHEMBL2079606)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  0.600nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003200(CHEMBL267849 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.600nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003201(CHEMBL386376 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.910nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003667(4-{2-Acetylamino-2-[1-({[1-{1-[2-carbamoyl-1-(1-ca...)
Affinity DataIC50:  1.40nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003196(CHEMBL433647 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003202(CHEMBL331408 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  2.10nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003664(4-{2-Acetylamino-2-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataIC50:  2.40nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406489(CHEMBL2079549)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003201(CHEMBL386376 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  2.70nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding toCholecystokinin type A receptor in rat pancreatic membrane...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406497(CHEMBL2079606)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011545(CHEMBL430906 | Desamino-Tyr(SO3H)-Met-Gly-Trp-Met-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406690(CHEMBL2112635)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003200(CHEMBL267849 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003670(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  4.40nMAssay Description:Concentration of the compound inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011538(Ac-Phe(4-SO3H)-Met-Gly-Trp-Met-Asp-Phe-NH2 | CHEMB...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011538(Ac-Phe(4-SO3H)-Met-Gly-Trp-Met-Asp-Phe-NH2 | CHEMB...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003196(CHEMBL433647 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  4.90nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011541(3-4-(tetrazol-5-ylphenyl)propanoyl-Met-Gly-Trp-Met...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003207(CHEMBL405805 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  5.5nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003662(4-{2-Acetylamino-2-[1-({[1-{1-[2-(1-carbamoyl-2-ph...)
Affinity DataIC50:  8.30nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003205(CHEMBL421471 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003203(CHEMBL436199 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406496(CHEMBL2079551)
Affinity DataIC50:  18nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406490(CHEMBL2079603)
Affinity DataIC50:  21nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003205(CHEMBL421471 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  22nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011542(3-[4-(carboxymethyl)phenyl]propanoyl-Met-Gly-Trp-M...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003665(3-{2-[2-(2-{2-[2-Acetylamino-3-(4-sulfo-phenyl)-pr...)
Affinity DataIC50:  22nMAssay Description:Concentration inhibiting [3H]-propanoyl-CCK-8 binding to cholecystokinin type B receptor of bovine striatum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011544(Ac-(R,S)Phe(3-CH2COOH)-Met-Gly-Trp-Met-Asp-Phe-NH2...)
Affinity DataIC50:  23nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011544(Ac-(R,S)Phe(3-CH2COOH)-Met-Gly-Trp-Met-Asp-Phe-NH2...)
Affinity DataIC50:  23nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003204(CHEMBL122438 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  25nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011542(3-[4-(carboxymethyl)phenyl]propanoyl-Met-Gly-Trp-M...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406491(CHEMBL2079548)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011541(3-4-(tetrazol-5-ylphenyl)propanoyl-Met-Gly-Trp-Met...)
Affinity DataIC50:  35nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406489(CHEMBL2079549)
Affinity DataIC50:  54nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003668(CHEMBL3143146 | [1-[1-[4-(1-Carbamoyl-2-phenyl-eth...)
Affinity DataIC50:  59nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406491(CHEMBL2079548)
Affinity DataIC50:  62nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406492(CHEMBL2079601)
Affinity DataIC50:  62nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406496(CHEMBL2079551)
Affinity DataIC50:  67nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406493(CHEMBL2079604)
Affinity DataIC50:  68nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003207(CHEMBL405805 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  73nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406495(CHEMBL2079547)
Affinity DataIC50:  76nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406488(CHEMBL2079550)
Affinity DataIC50:  92nMAssay Description:Inhibition of [3H]-propanoyl binding to cholecystokinin type B receptor subtype was determined in bovine striatum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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