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Found 20 with Last Name = 'michelson' and Initial = 'rh'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92983(MPP analogue, 19)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92982(MPP analogue, 18)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92981(MPP analogue, 17)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50018078(2-(4-Phenyl-piperidin-1-yl)-cyclohexanol | 2-(4-Ph...)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  36nMAssay Description:Displacement of [3H]vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009603(1-(3-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009597(1-(3-Iodo-phenyl)-3-(4-phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50:  73nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009604(1-(3-Methoxy-phenyl)-3-(4-phenyl-piperidin-1-yl)-p...)
Affinity DataIC50:  115nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009600(1-Naphthalen-2-yl-3-(4-phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50:  145nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009599(4-[2-Hydroxy-3-(4-phenyl-piperidin-1-yl)-propyl]-p...)
Affinity DataIC50:  220nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  328nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009595(1-(4-Bromo-phenyl)-3-(4-phenyl-piperidin-1-yl)-pro...)
Affinity DataIC50:  328nMAssay Description:Displacement of [3H]vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009598(3-[2-Hydroxy-3-(4-phenyl-piperidin-1-yl)-propyl]-p...)
Affinity DataIC50:  520nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009601(1-(3-Bromo-phenyl)-3-(4-phenyl-piperazin-1-yl)-pro...)
Affinity DataIC50:  990nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009596(1-Naphthalen-1-yl-3-(4-phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Torpedo californica)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50009594(1-(4-Bromo-phenyl)-3-(4-phenyl-piperazin-1-yl)-pro...)
Affinity DataIC50:  1.54E+3nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92981(MPP analogue, 17)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92983(MPP analogue, 19)
Affinity DataIC50:  8.50E+5nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University of California San Francisco

LigandPNGBDBM92982(MPP analogue, 18)
Affinity DataIC50:  2.00E+6nMAssay Description:Inhibition assay using MAO-A and MAO-B.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed