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Found 137 with Last Name = 'mihm' and Initial = 'g'
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043257(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl-1-[...)
Affinity DataIC50:  3nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043260(2-Butyl-6-(1,1-dioxo-1lambda*6*-[1,2]thiazinan-2-y...)
Affinity DataIC50:  3nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043244(4'-(1-Methyl-2'-propyl-1H-[2,5']bibenzoimidazolyl-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataIC50:  3nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043277(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50:  4nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043246(4'-(6-Imidazo[1,2-a]pyridin-2-yl-4-methyl-2-propyl...)
Affinity DataIC50:  4nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129977(4-[7-(1,1-Dimethyl-2-oxo-2-pyrrolidin-1-yl-ethyl)-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043247(4-Methyl-2-propyl-6-pyridin-2-yl-1-[2'-(1H-tetrazo...)
Affinity DataIC50:  5nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043279(1-Methyl-2'-propyl-3'-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50:  5nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129957(2-[2-(4-Carbamimidoyl-phenoxy)-4-methyl-quinolin-7...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129976(4-{4-Methyl-3-oxo-7-[1-(pyrrolidine-1-carbonyl)-cy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043248(3-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50:  8nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129968(4-[7-(1,1-Dimethyl-2-oxo-2-piperidin-1-yl-ethyl)-4...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043263(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50:  10nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129973(2-[3-(4-Carbamimidoyl-benzyl)-1-methyl-2-oxo-1,2-d...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043255(2-Propyl-6-pyridin-2-yl-1-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50:  11nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129979(4-{7-[1,1-Dimethyl-2-(3-methyl-piperidin-1-yl)-2-o...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129974(4-{7-[1-(2-Hydroxymethyl-pyrrolidine-1-carbonyl)-c...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043271(1,7'-Dimethyl-2'-propyl-3'-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129969(CHEMBL74263 | N-{1-[3-(4-Carbamimidoyl-benzyl)-1-m...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129972(2-[3-(4-Carbamimidoyl-benzyl)-1-methyl-2-oxo-1,2-d...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043252(1-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50:  21nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043269(4'-[2-Butyl-6-(3,3-dimethyl-ureido)-benzoimidazol-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50035429(4'-[2-Butyl-6-(3-cyclohexyl-ureido)-benzoimidazol-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043268(4'-[2-Butyl-6-(3-cyclohexyl-1-methyl-ureido)-benzo...)
Affinity DataIC50:  26nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129970(1-[3-(4-Carbamimidoyl-benzyl)-1-methyl-2-oxo-1,2-d...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129964(1-[2-(4-Carbamimidoyl-phenoxy)-4-methyl-quinolin-7...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018292(11-[2-(2-Diethylaminomethyl-piperidin-1-yl)-acetyl...)
Affinity DataIC50:  30nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018304(11-(2-{2-[(Cycloheptyl-methyl-amino)-methyl]-piper...)
Affinity DataIC50:  30nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043281(4'-{2-Butyl-6-[methyl-(propane-1-sulfonyl)-amino]-...)
Affinity DataIC50:  33nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043249(4'-[2-Butyl-6-(1,1-dioxo-1lambda*6*-[1,2]thiazinan...)
Affinity DataIC50:  34nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  35nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018302(9-Chloro-11-[2-(2-diethylaminomethyl-piperidin-1-y...)
Affinity DataIC50:  40nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018291(11-{2-[2-(3-Diethylamino-propyl)-piperidin-1-yl]-a...)
Affinity DataIC50:  60nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018314(11-(2-{2-[(Cyclohexyl-methyl-amino)-methyl]-piperi...)
Affinity DataIC50:  60nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129975(4-[7-(1,1-Dimethyl-2-oxo-2-piperazin-1-yl-ethyl)-4...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018294(11-[2-(2-Diethylaminomethyl-piperidin-1-yl)-acetyl...)
Affinity DataIC50:  70nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018304(11-(2-{2-[(Cycloheptyl-methyl-amino)-methyl]-piper...)
Affinity DataIC50:  70nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043270(4'-[2-Butyl-6-(2-oxo-piperidin-1-yl)-benzoimidazol...)
Affinity DataIC50:  81nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50129976(4-{4-Methyl-3-oxo-7-[1-(pyrrolidine-1-carbonyl)-cy...)
Affinity DataIC50:  84nMAssay Description:Inhibition of coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043265(4'-(2-Butyl-6-pentanoylamino-benzoimidazol-1-ylmet...)
Affinity DataIC50:  86nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018298(11-(2-{2-[(Butyl-methyl-amino)-methyl]-piperidin-1...)
Affinity DataIC50:  100nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018306(8-Chloro-11-[2-(2-diethylaminomethyl-piperidin-1-y...)
Affinity DataIC50:  100nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018293(11-(2-{2-[(Ethyl-methyl-amino)-methyl]-piperidin-1...)
Affinity DataIC50:  120nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018297(11-[2-(2-Dimethylaminomethyl-piperidin-1-yl)-acety...)
Affinity DataIC50:  140nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataIC50:  140nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018305(8-Bromo-11-[2-(2-diethylaminomethyl-piperidin-1-yl...)
Affinity DataIC50:  150nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018314(11-(2-{2-[(Cyclohexyl-methyl-amino)-methyl]-piperi...)
Affinity DataIC50:  150nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50018299(11-[2-(2-Diethylaminomethyl-pyrrolidin-1-yl)-acety...)
Affinity DataIC50:  150nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043275(4'-(6-Dimethylaminomethyl-4-methyl-2-propyl-benzoi...)
Affinity DataIC50:  158nMAssay Description:Inhibition of specific binding of [125I]-angiotensin-II to angiotensin 1 receptor in rat lung membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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