Compile Data Set for Download or QSAR
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Found 93 with Last Name = 'miles' and Initial = 't'
TargetAurora kinase B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  40nMAssay Description:Inhibition of aurora B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  63nMAssay Description:Inhibition of CB1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50548060(CHEMBL4762609)
Affinity DataIC50:  110nMAssay Description:Inhibition of human ERK8 (2 to 544 residues) incubated for 5 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)
Affinity DataIC50:  114nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50384600(CHEMBL2036792 | US9744172, Compound UNC00000563A)
Affinity DataIC50:  199nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  500nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50548060(CHEMBL4762609)
Affinity DataIC50:  550nMAssay Description:Inhibition of human p38beta MAPK (1 to 364 residues) incubated for 5 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359538(CHEMBL1235773)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359457(CHEMBL1926867)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359535(CHEMBL1927163)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50463653(CHEMBL4241707)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50542902(CHEMBL4645906)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of MAOA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359544(CHEMBL1927168)
Affinity DataIC50:  4.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613723(CHEMBL5268330)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359536(CHEMBL1927165)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50463654(CHEMBL4241692)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613719(CHEMBL5281165)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359541(CHEMBL1927162)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells by patch-clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated for 20 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613721(CHEMBL5275547)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359537(CHEMBL1927167)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359542(CHEMBL1927164)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol 14-alpha demethylase(Trypanosoma cruzi)
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50463655(CHEMBL546608 | TCMDC-124726)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi CYP51More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))TBA
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50357934(CHEMBL1916532)
Affinity DataIC50:  1.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50493332(CHEMBL2424930)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50517286(CHEMBL4516798)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613720(CHEMBL5283073)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human CDK4 by kinobeads-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613716(CHEMBL5283476)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613725(CHEMBL5268278)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359451(CHEMBL1926763)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359452(CHEMBL1926765)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359450(CHEMBL1926762)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359540(CHEMBL1927161)
Affinity DataIC50:  2.51E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359454(CHEMBL1926864)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human ERG by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50359545(CHEMBL1927170)
Affinity DataIC50:  2.95E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613726(CHEMBL5272922)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50517287(CHEMBL4563818)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50517285(CHEMBL4572962)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50613718(CHEMBL5286709)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERG potassium channel by Q-patch clamp assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAurora kinase B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50601512(DDD-01305143 | DDD01305143 | GSK-3494245 | GSK3494...)
Affinity DataIC50: <3.16E+4nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
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