Compile Data Set for Download or QSAR
maximum 50k data
Found 132 with Last Name = 'minnicozzi' and Initial = 'm'
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211457(3-(2-((R)-1-(4-sec-butylfuran-2-yl)propylamino)-3,...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211449((R)-3-(3,4-dioxo-2-(1-(4-(pentan-3-yl)furan-2-yl)p...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211454((R)-3-(2-(1-(4-ethylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211458((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)propy...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211456((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)ethyl...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211453((R)-3-(2-(1-(4-butylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211458((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)propy...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211462((R)-3-(2-(cyclopropyl(4-isopropylfuran-2-yl)methyl...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211450((R)-3-(2-(1-(4-cyclopentylfuran-2-yl)propylamino)-...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211464((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-methylfuran-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211448((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)-2,2-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211452((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)-2-me...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211459((R)-3-(2-(1-(4-cyclohexylfuran-2-yl)propylamino)-3...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211455((R)-3-(2-(1-(4-tert-butylfuran-2-yl)propylamino)-3...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50200877((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylthioph...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50200880((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211451((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-methylthioph...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211463((S)-3-(3,4-dioxo-2-(2,2,2-trifluoro-1-(4-isopropyl...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211454((R)-3-(2-(1-(4-ethylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211457(3-(2-((R)-1-(4-sec-butylfuran-2-yl)propylamino)-3,...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211464((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-methylfuran-...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211461((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-(4-morpholin...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211460((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(3-methylthioph...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211455((R)-3-(2-(1-(4-tert-butylfuran-2-yl)propylamino)-3...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211462((R)-3-(2-(cyclopropyl(4-isopropylfuran-2-yl)methyl...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211452((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)-2-me...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211448((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)-2,2-...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211461((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-(4-morpholin...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211463((S)-3-(3,4-dioxo-2-(2,2,2-trifluoro-1-(4-isopropyl...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50200880((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211451((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(4-methylthioph...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211465((R)-3-(2-(1-(3-ethylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211449((R)-3-(3,4-dioxo-2-(1-(4-(pentan-3-yl)furan-2-yl)p...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211453((R)-3-(2-(1-(4-butylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211456((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)ethyl...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211450((R)-3-(2-(1-(4-cyclopentylfuran-2-yl)propylamino)-...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211460((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(3-methylthioph...)
Affinity DataKi:  123nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50200877((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylthioph...)
Affinity DataKi:  146nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211459((R)-3-(2-(1-(4-cyclohexylfuran-2-yl)propylamino)-3...)
Affinity DataKi:  283nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211465((R)-3-(2-(1-(3-ethylfuran-2-yl)propylamino)-3,4-di...)
Affinity DataKi:  379nMAssay Description:Displacement of [125I]IL8 from human CXCR1 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219278(CHEMBL250137 | [5-aminomethyl-2-(8-methoxy-2-trifl...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219274(8-[5-aminomethyl-2-(8-methoxy-2-trifluoromethyl-qu...)
Affinity DataIC50:  1nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219281(CHEMBL399385 | [5-aminomethyl-2-(8-methoxy-2-trifl...)
Affinity DataIC50:  1nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219277(4-(5-(aminomethyl)-2-(8-methoxy-2-(trifluoromethyl...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211458((R)-2-hydroxy-3-(2-(1-(4-isopropylfuran-2-yl)propy...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [125I]IL8 from human CXCR2 expressed in CHO cells by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219268(CHEMBL399298 | tert-butyl (R)-1-(5-(aminomethyl)-2...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219273((Z)-(5-(aminomethyl)-2-(8-methoxy-2-(trifluorometh...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219272((5-(aminomethyl)-2-(8-methoxy-2-(trifluoromethyl)q...)
Affinity DataIC50:  2nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219269((5-(aminomethyl)-2-(8-methoxy-2-(trifluoromethyl)q...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50219275(CHEMBL249691 | tert-butyl 4-(5-(aminomethyl)-2-(8-...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of PDE4BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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