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Found 119 with Last Name = 'misura' and Initial = 'as'
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211814(4-(2-(4-fluorophenyl)-7-((isopropylamino)methyl)H-...)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211811(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374578(CHEMBL401749)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211805(4-(7-(((3-(dimethylamino)propyl)(methyl)amino)meth...)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374594(CHEMBL444009)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182359(CHEMBL379059 | N-benzyl-4-(7-((dimethylamino)methy...)
Affinity DataIC50:  0.0810nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211820(4-(7-(((2-(azetidin-1-yl)ethyl)(methyl)amino)methy...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211812(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211802(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211803(4-(7-((ethyl(methyl)amino)methyl)-2-(4-fluoropheny...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211808(CHEMBL233008 | N-(2-(((2-(4-fluorophenyl)-3-(2-((S...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211821(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171694((R)-5-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.160nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374591(CHEMBL255128)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374587(CHEMBL272573)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211819(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211816((S)-2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethy...)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374588(CHEMBL255381)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211810(4-(2-(4-fluorophenyl)-7-((methyl((tetrahydrofuran-...)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50182361(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374592(CHEMBL271922)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211823(4-(7-((ethyl(methyl)amino)methyl)-2-(4-fluoropheny...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211818(CHEMBL233011 | N-tert-butyl-4-(7-((dimethylamino)m...)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374580(CHEMBL271638)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50183915((5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-y...)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374590(CHEMBL406910)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171685(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.380nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211822(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50:  0.390nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374593(CHEMBL429745)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171698(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171707(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.410nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211817(4-(7-(azetidin-1-ylmethyl)-2-(4-fluorophenyl)H-imi...)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171705(1-Benzyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171699((S)-1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168176(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.530nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171695((R)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyr...)
Affinity DataIC50:  0.560nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211815(1-(azetidin-1-yl)-2-(((2-(4-fluorophenyl)-3-(2-((S...)
Affinity DataIC50:  0.570nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171688(1-Ethoxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50211806(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171702(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374585(CHEMBL255631)
Affinity DataIC50:  0.670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171690(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.690nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171695((R)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyr...)
Affinity DataIC50:  0.690nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171692(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.710nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168193(2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.710nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.710nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50183909(1-(5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2...)
Affinity DataIC50:  0.710nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171686(1-Allyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-y...)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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