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Found 120 with Last Name = 'miyashita' and Initial = 'h'
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189833((S)-N-butyl-3-((S)-2-(4-fluorophenylsulfonamido)-3...)
Affinity DataIC50:  21nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189833((S)-N-butyl-3-((S)-2-(4-fluorophenylsulfonamido)-3...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)
Affinity DataIC50:  49nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189828(1-((S)-1-((3S)-2-hydroxy-tetrahydrofuran-3-ylamino...)
Affinity DataIC50:  86nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189825((2S)-2-((((4-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189825((2S)-2-((((4-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189835((2S)-2-((((4-fluorophenyl)amino)thioxomethyl)amino...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189822((2S)-2-((benzylamino)thioxomethyl)amino)-4-methyl-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189834((2S)-2-((((3-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  170nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189832((2S)-4-methyl-2-((((4-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  170nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189831((2S)-4-methyl-2-((((3-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189835((2S)-2-((((4-fluorophenyl)amino)thioxomethyl)amino...)
Affinity DataIC50:  190nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189828(1-((S)-1-((3S)-2-hydroxy-tetrahydrofuran-3-ylamino...)
Affinity DataIC50:  190nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189827((2S)-2-((((4-methoxyphenyl)amino)thioxomethyl)amin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189827((2S)-2-((((4-methoxyphenyl)amino)thioxomethyl)amin...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189830((2S)-4-methyl-2-((((2-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189822((2S)-2-((benzylamino)thioxomethyl)amino)-4-methyl-...)
Affinity DataIC50:  240nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189830((2S)-4-methyl-2-((((2-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  250nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189834((2S)-2-((((3-cyanophenyl)amino)thioxomethyl)amino)...)
Affinity DataIC50:  260nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189831((2S)-4-methyl-2-((((3-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  340nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114342((E)-2-(dimethylamino)-N'-((S)-2-((S)-2-(4-fluoroph...)
Affinity DataIC50:  370nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189823((2S,3S)-3-methyl-2-(((phenylamino)thioxomethyl)ami...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189829((2S)-3-methyl-2-(((phenylamino)thioxomethyl)amino)...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189826((S)-2-(4-fluorophenylsulfonamido)-N-((3S)-2-hydrox...)
Affinity DataIC50:  880nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189832((2S)-4-methyl-2-((((4-methylphenyl)amino)thioxomet...)
Affinity DataIC50:  910nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53408((2S)-2-[[5-(3,4-dihydro-1H-isoquinoline-2-carbonyl...)
Affinity DataIC50: >1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53402((3R,3aR,7aR)-2-benzyl-3-(1-bromo-2-naphthyl)-7a-me...)
Affinity DataIC50:  1.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189823((2S,3S)-3-methyl-2-(((phenylamino)thioxomethyl)ami...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189829((2S)-3-methyl-2-(((phenylamino)thioxomethyl)amino)...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53401((3R,3aS,7R,7aS)-2-benzyl-3-(3-chloro-4-methoxy-phe...)
Affinity DataIC50:  2.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53412(4-[[5-[[(1S)-1-tert-butoxycarbonyl-5-(tert-butoxyc...)
Affinity DataIC50:  2.50E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189826((S)-2-(4-fluorophenylsulfonamido)-N-((3S)-2-hydrox...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53404((3R,3aR,7aR)-2-benzyl-3-[4-fluoro-3-(4-methylpheny...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53405(4-(4-methoxyphenyl)-5,8-dimethyl-2-phenyl-3,4-dihy...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53403((3R,3aR,7aR)-2-benzyl-3-(5-bromo-2-methoxy-phenyl)...)
Affinity DataIC50:  5.00E+3nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM16415((1,3-dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)acetic...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53406((6Z)-1-benzoyl-4-(4-fluorobenzyl)-5-(4-methoxyphen...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53409((2S)-2-[[4-[[(1S)-2-tert-butoxy-2-keto-1-methyl-et...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53410(4-[[5-[[(1S)-1-benzyl-2-tert-butoxy-2-keto-ethyl]c...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53411((2S)-2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imida...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase ESS1(Saccharomyces cerevisiae (Baker's yeast))
Tohoku University

LigandPNGBDBM53407(2-(2-methoxyphenyl)-8-nitro-5-oxidanyl-chromen-4-o...)
Affinity DataIC50: >1.00E+4nMpH: 7.0 T: 2°CAssay Description:Assay was carried out measuring the MCA fluorescence using Suc-Ala-Glu-Pro-Phe-MCA as substrate purchased from Japan Peptide Institute Co.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Sus scrofa)
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189824(CHEMBL206737 | N-(1-cyano-3-methylbutyl)-2-((4-flu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of porcein kidney m calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Senju Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50189824(CHEMBL206737 | N-(1-cyano-3-methylbutyl)-2-((4-flu...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human erythrocyte mu calpainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446690(CHEMBL3113624)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446691(CHEMBL3113623)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446692(CHEMBL3113622)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446693(CHEMBL3113843)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446696(CHEMBL3113840)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50446697(CHEMBL3113839)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human GPR119 transfected in CHO cells assessed as cAMP accumulation after 2 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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