Found 417 with Last Name = 'mock' and Initial = 'ed' TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 2(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT2 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of trypsin-like activity of proteasome in human NCI-H929 cells after 6 hrs by proteasomeGlo assayMore data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 4(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT4 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 4(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT4 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta 5 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta 5 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr...More data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of trypsin-like activity of proteasome in human NCI-H929 cells after 6 hrs by proteasomeGlo assayMore data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 155nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 2(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT2 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta 5 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of trypsin-like activity of proteasome in human RPMI-8226 cells after 6 hrs by proteasomeGlo assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of trypsin-like activity of proteasome in human NCI-H929 cells after 6 hrs by proteasomeGlo assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of trypsin-like activity of proteasome beta 2 subunit in HEK-293T cell lysates using BODIPY-BODIPY-TMR-epoxomicin as probe after 1 hr by S...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 4(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT4 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 4(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT4 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 2(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT2 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 3(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT3 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetPhospholipase A and acyltransferase 5(Homo sapiens)
Leiden University & Oncode Institute
Curated by ChEMBL
Leiden University & Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of full-length C-terminal FLAG-tagged human PLAAT5 expressed in HEK293T cell lysate preincubated for 30 mins followed by MB064 addition an...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Leiden Institute Of Chemistry And Netherlands Proteomics Centre
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of trypsin-like activity of proteasome in human NCI-H929 cells after 6 hrs by proteasomeGlo assayMore data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 209nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
TargetN-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D(Homo sapiens)
Leiden University And Oncode Institute
Curated by ChEMBL
Leiden University And Oncode Institute
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Inhibition of full length human NAPE-PLD expressed in HEK293T cell lysate using PED6 as substrate preincubated for 30 mins followed by substrate addi...More data for this Ligand-Target Pair
