Affinity DataKi: 0.339nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.871nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.17nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.32nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.74nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.86nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.95nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.19nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Competitive inhibition of N-terminal His6-tagged KDM4C (1 to 352 residues) (unknown origin) expressed in Escherichia coli Rosetta 2(DE3)pLysS using A...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-DTG from the Sigma2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.57nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.82nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.39nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.89nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.47nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.13nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.75nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.17nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.61nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.76nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.41nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.32nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.51nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 9.12nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.33nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Qbi Covid-19 Research Group (Qcrg)
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-pentazocin from the Sigma1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair