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Found 244 with Last Name = 'morse' and Initial = 'em'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50210164(CHEMBL2132936)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]-Nalpha-methylhistamine binding to H3 receptor in guinea-pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348384(CHEMBL1800383)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348373(CHEMBL1800373)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348393(CHEMBL1800246)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of recombinant HDAC9 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348376(CHEMBL1800375)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348397(CHEMBL1800250)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of recombinant HDAC3 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of recombinant HDAC1 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348393(CHEMBL1800246)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM55151(1-(3,4-Dihydroxy-phenyl)-2-(4-hydroxy-6-methyl-pyr...)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of recombinant HDAC2 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of recombinant HDAC8 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of recombinant HDAC7 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348380(CHEMBL1800379)
Affinity DataIC50:  2.48E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  2.79E+4nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348393(CHEMBL1800246)
Affinity DataIC50:  3.19E+4nMAssay Description:Inhibition of recombinant HDAC7 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  3.25E+4nMAssay Description:Inhibition of recombinant HDAC4 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348379(CHEMBL1800378)
Affinity DataIC50:  3.26E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348384(CHEMBL1800383)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of recombinant HDAC3 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348377(CHEMBL1800376)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348384(CHEMBL1800383)
Affinity DataIC50:  4.86E+4nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348393(CHEMBL1800246)
Affinity DataIC50:  5.42E+4nMAssay Description:Inhibition of recombinant HDAC4 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348374(CHEMBL1307946)
Affinity DataIC50:  6.09E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348376(CHEMBL1800375)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of recombinant HDAC2 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348384(CHEMBL1800383)
Affinity DataIC50:  6.93E+4nMAssay Description:Inhibition of recombinant HDAC2 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348388(CHEMBL1800241)
Affinity DataIC50:  7.41E+4nMAssay Description:Inhibition of recombinant HDAC9 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348384(CHEMBL1800383)
Affinity DataIC50:  7.72E+4nMAssay Description:Inhibition of recombinant HDAC1 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348376(CHEMBL1800375)
Affinity DataIC50:  8.23E+4nMAssay Description:Inhibition of recombinant HDAC1 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348376(CHEMBL1800375)
Affinity DataIC50:  8.64E+4nMAssay Description:Inhibition of recombinant HDAC3 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348393(CHEMBL1800246)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition of recombinant HDAC6 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348375(CHEMBL1800374)
Affinity DataIC50:  9.43E+4nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348387(CHEMBL1800385)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348390(CHEMBL1800243)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348391(CHEMBL1800244)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348392(CHEMBL1800245)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348382(CHEMBL1800381)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348383(CHEMBL1800382)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348385(CHEMBL1800384)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348389(CHEMBL1800242)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348378(CHEMBL1800377)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348379(CHEMBL1800378)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348380(CHEMBL1800379)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM96613(2-[(4-keto-6-methyl-1H-pyrimidin-2-yl)thio]-N-phen...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348381(CHEMBL1800380)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM55151(1-(3,4-Dihydroxy-phenyl)-2-(4-hydroxy-6-methyl-pyr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348376(CHEMBL1800375)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348397(CHEMBL1800250)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348372(CHEMBL1800251)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Broad Institute Of Harvard And Mit

Curated by ChEMBL
LigandPNGBDBM50348373(CHEMBL1800373)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant HDAC5 assessed as inhibition of fluorogenic aminocoumarin release from substrate by trypsin-coupled biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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