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Found 283 with Last Name = 'mullen' and Initial = 'd'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030062(Ac-(D-Pen)-I-P-R-G-D-(Y-OMe)-R-C-NH2 | CHEMBL43846...)
Affinity DataIC50:  2nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030068(Ac-C-I-P-R-G-D-Y-R-C-NH2 | CHEMBL405541)
Affinity DataIC50:  3nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030050(Ac-C-I-P-R-G-D-(Y-OMe)R-C-NH2 | CHEMBL429529)
Affinity DataIC50:  3nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030066(Ac-C-N-P-R-G-D-(Y-OMe)-O-C-NH2 | CHEMBL2371530)
Affinity DataIC50:  6nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030066(Ac-C-N-P-R-G-D-(Y-OMe)-O-C-NH2 | CHEMBL2371530)
Affinity DataIC50:  6nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030066(Ac-C-N-P-R-G-D-(Y-OMe)-O-C-NH2 | CHEMBL2371530)
Affinity DataIC50:  6nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030057(CHEMBL2371489 | R(Pmc)-G-(DH)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  10nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030069(CHEMBL2371473 | R(Pmc)-G-H-R-G-D-(p-I-F)-R-C-R)
Affinity DataIC50:  10nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030069(CHEMBL2371473 | R(Pmc)-G-H-R-G-D-(p-I-F)-R-C-R)
Affinity DataIC50:  10nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030069(CHEMBL2371473 | R(Pmc)-G-H-R-G-D-(p-I-F)-R-C-R)
Affinity DataIC50:  10nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030057(CHEMBL2371489 | R(Pmc)-G-(DH)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  10nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030064(Ac-C-I-P-R-G-D-F-R-C-NH2 | CHEMBL265425)
Affinity DataIC50:  14nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030059(Ac-C-I-P-R-G-D-(Y-O-n-butyl)-R-C-NH2 | CHEMBL40887...)
Affinity DataIC50:  16nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030033(CHEMBL2371524 | R(Pmc)-G-Y-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  17nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030033(CHEMBL2371524 | R(Pmc)-G-Y-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  17nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030033(CHEMBL2371524 | R(Pmc)-G-Y-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  17nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)
Affinity DataIC50:  19nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030046((Pmc)-G-H-R-G-D-L-R-C-A | CHEMBL266826)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030070(CHEMBL2371527 | R(Pmc)-G-H-R-G-D-(Hpa)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030070(CHEMBL2371527 | R(Pmc)-G-H-R-G-D-(Hpa)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030049(CHEMBL2371472 | R(Pmc)-G-H-R-G-D-(p-Cl-F)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030070(CHEMBL2371527 | R(Pmc)-G-H-R-G-D-(Hpa)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030049(CHEMBL2371472 | R(Pmc)-G-H-R-G-D-(p-Cl-F)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305013(3-(2-amino-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol...)
Affinity DataIC50:  20nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030049(CHEMBL2371472 | R(Pmc)-G-H-R-G-D-(p-Cl-F)-R-C-R)
Affinity DataIC50:  20nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030052(CHEMBL2371480 | R(Pmc)-G-(DY)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  30nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030052(CHEMBL2371480 | R(Pmc)-G-(DY)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  30nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030052(CHEMBL2371480 | R(Pmc)-G-(DY)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  30nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030052(CHEMBL2371480 | R(Pmc)-G-(DY)-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  30nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)
Affinity DataIC50:  33nMAssay Description:Inhibition of IKK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305007(5-(3-aminopropyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-...)
Affinity DataIC50:  35nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50227629(CHEMBL433084)
Affinity DataIC50:  36nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305010(3-(2-amino-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol...)
Affinity DataIC50:  37nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030032(Ac-C-N-P-R-G-D-(Y-OMe)-K-C-NH2 | CHEMBL267950)
Affinity DataIC50:  38nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030030(CHEMBL2371540 | R(Pen)-G-H-R-G-D-L-R-C-R)
Affinity DataIC50:  40nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030047(CHEMBL2371477 | R(Pmc)-G-H-R-G-D-F-R-C-R)
Affinity DataIC50:  40nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030030(CHEMBL2371540 | R(Pen)-G-H-R-G-D-L-R-C-R)
Affinity DataIC50:  40nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030047(CHEMBL2371477 | R(Pmc)-G-H-R-G-D-F-R-C-R)
Affinity DataIC50:  40nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030047(CHEMBL2371477 | R(Pmc)-G-H-R-G-D-F-R-C-R)
Affinity DataIC50:  40nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305014(3-(2-amino-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol...)
Affinity DataIC50:  41nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)
Affinity DataIC50:  44nMAssay Description:Inhibition of CHK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)
Affinity DataIC50:  53nMAssay Description:Inhibition of pdk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305003(7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-p...)
Affinity DataIC50:  56nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030048(CHEMBL2371529 | R(Pmc)-I-H-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  60nMAssay Description:Binding affinity against integrin alpha 2b-beta 3 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030048(CHEMBL2371529 | R(Pmc)-I-H-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  60nMAssay Description:Binding affinity against integrin alpha V-beta5 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
Telios Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030048(CHEMBL2371529 | R(Pmc)-I-H-R-G-D-(Y-OMe)-R-C-R)
Affinity DataIC50:  60nMAssay Description:Binding affinity against integrin alpha5-beta1 in enzyme linked immunosorbent assay (ELISA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50227633(CHEMBL296753)
Affinity DataIC50:  83nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50227634(CHEMBL48617)
Affinity DataIC50:  90nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50227630(CHEMBL49309)
Affinity DataIC50:  96nMAssay Description:Ability to inhibit binding of titreated serotonin to the 5-hydroxytryptamine 1 receptor in rat brain frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50305006(5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-i...)
Affinity DataIC50:  98nMAssay Description:Inhibition of PKCetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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