Compile Data Set for Download or QSAR
maximum 50k data
Found 13 with Last Name = 'murruzzu' and Initial = 'c'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50216315((1R,4R)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[...)
Affinity DataKi:  0.0180nMAssay Description:Displacement of [3H]cytosine form alpha4beta2 nAChR in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275878(3-(6-chloropyridin-3-yl)-3,6-diazabicyclo[3.1.1]he...)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275880(3-(6-bromopyridin-3-yl)-3,6-diazabicyclo[3.1.1]hep...)
Affinity DataKi:  0.0390nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275879(3-(pyridin-3-yl)-3,6-diazabicyclo[3.1.1]heptane | ...)
Affinity DataKi:  0.0560nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275932(3-(6-chloropyridazin-3-yl)-3,6-diazabicyclo[3.1.1]...)
Affinity DataKi:  0.168nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275933(3-(6-chloropyridin-3-yl)-6-methyl-3,6-diazabicyclo...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275931(3-(4-nitrophenyl)-3,6-diazabicyclo[3.1.1]heptane |...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275879(3-(pyridin-3-yl)-3,6-diazabicyclo[3.1.1]heptane | ...)
Affinity DataKi:  1.36nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275878(3-(6-chloropyridin-3-yl)-3,6-diazabicyclo[3.1.1]he...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275933(3-(6-chloropyridin-3-yl)-6-methyl-3,6-diazabicyclo...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275932(3-(6-chloropyridazin-3-yl)-3,6-diazabicyclo[3.1.1]...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275880(3-(6-bromopyridin-3-yl)-3,6-diazabicyclo[3.1.1]hep...)
Affinity DataKi:  50.5nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50275931(3-(4-nitrophenyl)-3,6-diazabicyclo[3.1.1]heptane |...)
Affinity DataKi:  2.80E+4nMAssay Description:Displacement of [3H]alpha-bungarotoxin form alpha7 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed