Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Binding affinity towards Melanocortin 1 receptor, expressed as negative log of the Ki valueMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Binding affinity towards Melanocortin 1 receptor, expressed as negative log of the Ki valueMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 1 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 1 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 1 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: 760nMAssay Description:Binding affinity towards Melanocortin 1 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 770nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Binding affinity towards Melanocortin 4 receptor using [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University
Curated by ChEMBL
Uppsala University
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair