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Found 142 with Last Name = 'nishimura' and Initial = 'k'
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50036731(3-Dimethylamino-1-phenyl-propan-1-one | CHEMBL5011...)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50047897(CHEMBL289199 | Dimethyl-(3-phenyl-propyl)-amine)
Affinity DataKi:  3.80E+5nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046768(2-Pentylamino-acetamide | 2-Pentylamino-acetamide(...)
Affinity DataKi:  9.40E+5nMAssay Description:Kinetic constant (KI) was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046768(2-Pentylamino-acetamide | 2-Pentylamino-acetamide(...)
Affinity DataKi:  1.08E+6nMAssay Description:Kinetic constant was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046767(CHEMBL344189 | Pentylamino-acetic acid ethyl ester)
Affinity DataKi:  2.00E+6nMAssay Description:Kinetic constant was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50047898(CHEMBL47794 | Dimethyl-pentyl-amine)
Affinity DataKi:  2.10E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50047896(CHEMBL46232 | Phenethyl-propyl-amine)
Affinity DataKi:  4.00E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046766(CHEMBL139751 | Pentylamino-acetonitrile)
Affinity DataKi:  4.94E+6nMAssay Description:Kinetic constant was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046769(3-Pentylamino-propionitrile | CHEMBL139492)
Affinity DataKi:  4.94E+6nMAssay Description:Kinetic constant was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046769(3-Pentylamino-propionitrile | CHEMBL139492)
Affinity DataKi:  5.79E+6nMAssay Description:Kinetic constant (KI) was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50018453(CHEMBL46278 | Dimethyl-phenethyl-amine | N,N-dimet...)
Affinity DataKi:  7.10E+6nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50016907(CHEMBL46841 | Dimethyl-(4-phenyl-butyl)-amine)
Affinity DataKi:  1.00E+7nMAssay Description:Inhibition of Monoamine oxidase-B from Bovine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046766(CHEMBL139751 | Pentylamino-acetonitrile)
Affinity DataKi:  1.40E+7nMAssay Description:Kinetic constant (KI) was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Bos taurus)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50046767(CHEMBL344189 | Pentylamino-acetic acid ethyl ester)
Affinity DataKi:  1.42E+7nMAssay Description:Kinetic constant (KI) was calculated by inhibition of monoamino oxidase B (MAO B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50287290(CHEMBL34866 | KRH-594 | Potassium; 2-[5-ethyl-3-[2...)
Affinity DataIC50:  0.440nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287294(2-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50:  0.440nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287291(CHEMBL35381 | N-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataIC50:  0.660nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107587(CHEMBL3601910)
Affinity DataIC50:  2.40nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50287289(2-Chloro-N-[5-ethyl-3-[2'-(1H-tetrazol-5-yl)-biphe...)
Affinity DataIC50:  3.60nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287292(CHEMBL34190 | Cyclopropanecarboxylic acid [5-ethyl...)
Affinity DataIC50:  6.5nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287295(CHEMBL35475 | N-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)-...)
Affinity DataIC50:  7.20nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107535(CHEMBL3601902)
Affinity DataIC50:  7.5nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107532(CHEMBL3601900)
Affinity DataIC50:  8.20nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107588(CHEMBL3601911)
Affinity DataIC50:  8.80nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107539(CHEMBL3601906)
Affinity DataIC50:  9.30nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107538(CHEMBL3601905)
Affinity DataIC50:  9.70nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50406795(Cozaar | LOSARTAN POTASSIUM)
Affinity DataIC50:  9.80nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107424(CHEMBL3600421)
Affinity DataIC50:  10nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107429(CHEMBL3600427)
Affinity DataIC50:  13nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107428(CHEMBL3600426)
Affinity DataIC50:  13nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50023929(CHEMBL3325502)
Affinity DataIC50:  15nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107452(CHEMBL3601898)
Affinity DataIC50:  15nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107585(CHEMBL3601908)
Affinity DataIC50:  17nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(Musca domestica)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107426(CHEMBL3600424)
Affinity DataIC50:  23nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107422(CHEMBL3601915)
Affinity DataIC50:  28nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107435(CHEMBL3600433)
Affinity DataIC50:  29nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107423(CHEMBL3600420)
Affinity DataIC50:  31nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107534(CHEMBL3601901)
Affinity DataIC50:  31nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107537(CHEMBL3601904)
Affinity DataIC50:  31nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50084137(2-Methyl-6-(phenylethynyl)pyridine | 2-Methyl-6-ph...)
Affinity DataIC50:  32nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50287293(CHEMBL286537 | N-[5-Ethyl-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50:  37nMAssay Description:Compound was tested in vitro for the ability to displace the specific binding of [125I]-A II from receptors in rat liver membrane(type 1 receptor)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107586(CHEMBL3601909)
Affinity DataIC50:  38nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107425(CHEMBL3600423)
Affinity DataIC50:  42nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107431(CHEMBL3600430)
Affinity DataIC50:  44nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50023797(CHEMBL3325511)
Affinity DataIC50:  52nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107421(CHEMBL3601913)
Affinity DataIC50:  56nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107395(CHEMBL3601912)
Affinity DataIC50:  56nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50107430(CHEMBL3600429)
Affinity DataIC50:  60nMAssay Description:Negative allosteric modulator activity against human mGluR5 expressed in HEK293 cells assessed as inhibition of glutamate-induced inositol phosphate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50023926(CHEMBL3325505)
Affinity DataIC50:  62nMAssay Description:Inhibition of human GlyT2 transfected in HEK293 cells assessed as [3H]glycine uptake after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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