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Found 223 with Last Name = 'ohmori' and Initial = 'o'
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223939(6-(4-methoxybenzyl)-7-neopentyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  1nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223914(6-((4-(4-fluorophenyl)piperazin-1-yl)methyl)-7-neo...)
Affinity DataIC50:  1nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223935(CHEMBL399842 | N-(4-((2-cyano-7-neopentyl-7H-pyrro...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223921(6-(4-(benzo[d][1,3]dioxol-5-yl)benzyl)-7-neopentyl...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223915(6-benzyl-7-neopentyl-7H-pyrrolo[2,3-d]pyrimidine-2...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223925(6-(4-((4-methylpiperazin-1-yl)methyl)benzyl)-7-cyc...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223919(7-(2,2-dimethylpropyl)-6-[(5-fluoro-2-oxospiro[ind...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223910(6-(4-chlorobenzyl)-7-cyclohexyl-7H-pyrrolo[2,3-d]p...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223911(7-neopentyl-6-((pyridin-4-yloxy)methyl)-7H-pyrrolo...)
Affinity DataIC50:  3nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223920(6-(4-morpholinobenzyl)-7-cyclohexyl-7H-pyrrolo[2,3...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184049(3-(6-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50:  4nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223936(6-((5,5-dimethyl-2,4-dioxooxazolidin-3-yl)methyl)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223940(6-((4,5-dichloro-1H-imidazol-1-yl)methyl)-7-neopen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223941(6-(4-((diethylamino)methyl)benzyl)-7-cyclohexyl-7H...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223937(6-((1H-1,2,3-triazol-1-yl)methyl)-7-neopentyl-7H-p...)
Affinity DataIC50:  5nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223918(6-((1H-imidazol-1-yl)methyl)-7-neopentyl-7H-pyrrol...)
Affinity DataIC50:  6nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223923(6-benzyl-7-cyclohexyl-7H-pyrrolo[2,3-d]pyrimidine-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50312718(CHEMBL479527 | torcetrapib)
Affinity DataIC50:  18nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50348228(CHEMBL1800807)
Affinity DataIC50:  18nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124871(US8759365, 9-4 | US8759365, 9-5)
Affinity DataIC50:  21nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124882(US8759365, 6)
Affinity DataIC50:  23nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124884(US8759365, 16-2)
Affinity DataIC50:  25nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50183986(CHEMBL207084 | N-(2-aminoethyl)-3-(2-(3,4,5-trimet...)
Affinity DataIC50:  29nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124878(US8759365, 23-10)
Affinity DataIC50:  30nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124876(US8759365, 17)
Affinity DataIC50:  32nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124881(US8759365, 14)
Affinity DataIC50:  34nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50183989(3-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50:  35nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184028(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50:  37nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184034(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2,3-...)
Affinity DataIC50:  38nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184019(CHEMBL379837 | N-(2-(dimethylamino)ethyl)-3-(2-(3,...)
Affinity DataIC50:  38nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124875(US8759365, 16)
Affinity DataIC50:  39nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124868(US8759365, 9-1)
Affinity DataIC50:  41nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124867(US8759365, 7-6)
Affinity DataIC50:  46nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124865(US8759365, 6-2)
Affinity DataIC50:  47nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCathepsin K(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50223928(6-biphenyl-4-ylmethyl-7-cyclohexyl-7H-pyrrolo[2,3-...)
Affinity DataIC50:  47nMAssay Description:Inhibition of cathepsin K by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124883(US8759365, 9)
Affinity DataIC50:  53nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124871(US8759365, 9-4 | US8759365, 9-5)
Affinity DataIC50:  54nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184002(CHEMBL207961 | N-(3-(dimethylamino)propyl)-3-(2-(3...)
Affinity DataIC50:  54nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124869(US8759365, 9-2)
Affinity DataIC50:  59nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124866(US8759365, 7-4)
Affinity DataIC50:  60nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250371(CHEMBL4064793)
Affinity DataIC50:  60nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250366(CHEMBL4075773)
Affinity DataIC50:  62nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184035(CHEMBL207499 | N-isobutyl-3-(3-(2-(3,4,5-trimethox...)
Affinity DataIC50:  63nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50184000(2-(3-(2-(3,4,5-trimethoxyphenylamino)-7H-pyrrolo[2...)
Affinity DataIC50:  63nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124877(US8759365, 18)
Affinity DataIC50:  63nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124864(US8759365, 6-1)
Affinity DataIC50:  69nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124873(US8759365, 9-6)
Affinity DataIC50:  70nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124870(US8759365, 9-3)
Affinity DataIC50:  70nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50250363(CHEMBL4070653)
Affinity DataIC50:  71nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM124874(US8759365, 11)
Affinity DataIC50:  72nMpH: 7.4 T: 2°CAssay Description:CETP Activity Kit (#RB-RPAK) was purchased from Roar Biochemical, Inc. (New York, N.Y., USA). To each well of a 96-well NBS half-area plate (costar #...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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