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Found 24 with Last Name = 'okumura' and Initial = 'k'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067222(CHEMBL128906 | [6-(4-Carbamimidoyl-benzoylamino)-c...)
Affinity DataIC50:  0.0730nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067216(CHEMBL129877 | {6-[4-(Imino-morpholin-4-yl-methyl)...)
Affinity DataIC50:  0.0980nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067228(CHEMBL131823 | [7-(4-Carbamimidoyl-benzoylamino)-1...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067217(CHEMBL323649 | {(S)-6-[4-(Imino-morpholin-4-yl-met...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067220(CHEMBL130405 | {7-[4-(N-Propylcarbamimidoyl)-benzo...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067224(CHEMBL130437 | {6-[4-(N-Prop-2-ynylcarbamimidoyl)-...)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067218(CHEMBL130878 | {7-[4-(Imino-morpholin-4-yl-methyl)...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067223(CHEMBL130892 | {7-[4-(N-Prop-2-ynylcarbamimidoyl)-...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067227(CHEMBL128539 | {7-[4-(N-Furan-2-ylmethyl-carbamimi...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067230(CHEMBL131593 | {7-[4-(N-Allylcarbamimidoyl)-benzoy...)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Mitsui Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067226(CHEMBL335160 | {(R)-6-[4-(Imino-morpholin-4-yl-met...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of Fibronogen binding to Immobilized Human Fibrinogen Receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50390978(VALSPODAR)
Affinity DataIC50:  291nMAssay Description:TP_TRANSPORTER: inhibition of Doxorubicin transepithelial transport (basal to apical) (Doxorubicin: 0.8 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50390978(VALSPODAR)
Affinity DataIC50:  1.06E+3nMAssay Description:TP_TRANSPORTER: inhibition of Vinblastine transepithelial transport (basal to apical) (Vinblastine: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  3.66E+3nMAssay Description:TP_TRANSPORTER: inhibition of Doxorubicin transepithelial transport (basal to apical) (Digoxin: 0.8 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50101815(CHEBI:7550 | Nicardipine)
Affinity DataIC50:  4.54E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50318911(CHEMBL1085699 | manidipine)
Affinity DataIC50:  4.65E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50088385(Benidipine | Benidipine HCl)
Affinity DataIC50:  4.96E+3nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50088384(Barnidipine | Barnidipine HCl)
Affinity DataIC50:  1.26E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50420237(EFONIDIPINE | EFONIDIPINE HYDROCHLORIDE)
Affinity DataIC50:  1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50103634(CL-287389 | FK-235 | Nilvadipine | Nivadipine | SK...)
Affinity DataIC50:  1.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50101963(BAY-K-5552 | CHEBI:76917 | Nisoldipine | Sular)
Affinity DataIC50:  4.41E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50237611(BAY-E-5009 | Baypress | CHEBI:7582 | Nitrendipine)
Affinity DataIC50:  6.82E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50004704((+)-cis-Diltiazem | (2S,3S)-5-(2-(dimethylamino)et...)
Affinity DataIC50:  7.77E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kobe University

Curated by ChEMBL
LigandPNGBDBM50101817(Adalat | Adalat Cc | Afeditab Cr | BAY-A-1040 | CH...)
Affinity DataIC50:  4.72E+5nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 0.1 uM) in MDR1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed