TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.03E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.37E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.56E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.67E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.05E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.38E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.39E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 5.76E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 6.43E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 7.04E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 7.23E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 3 [N508S](Homo sapiens (Human))
Georgia State University
Curated by ChEMBL
Georgia State University
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of His6X-tagged PRMT3 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 8.36E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of His6X-tagged PRMT5 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Georgia State University
Curated by ChEMBL
Georgia State University
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of His6X-tagged PRMT6 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.84E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.54E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 8.49E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged CARM1 expressed in escherichia coli BL21(DE3) cells using using [14C]-S-adenosyl-L-methionine and histone H3 peptide after 8...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.61E+5nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.84E+5nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.92E+5nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
The University Of Georgia
Curated by ChEMBL
The University Of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.68E+5nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair