TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Biomedical Research Foundation Academy Of Athens (Brfaa)
Curated by ChEMBL
Biomedical Research Foundation Academy Of Athens (Brfaa)
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of PI3Kalpha catalytic domain (unknown origin) using PIP2 liposomes as substrate in presence of biotin-labeled PIP3 and GST-GRP1-PH by str...More data for this Ligand-Target Pair