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Found 180 with Last Name = 'parekh' and Initial = 't'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0800nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.0990nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.150nMAssay Description:Compound was tested for binding affinity against human Melatonin receptor type 1B in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.290nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.380nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290238(CHEMBL80736 | N-[2-(2-Ethoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  0.390nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290238(CHEMBL80736 | N-[2-(2-Ethoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290234(CHEMBL440692 | N-[2-(2-Hydroxy-7-methoxy-naphthale...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290239(CHEMBL78751 | N-{2-[2-(2-Hydroxy-ethoxy)-7-methoxy...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9690(SCH446211 (SCH6) Analog 23 | tert-butyl N-[(2S)-1-...)
Affinity DataKi:  2nM ΔG°:  -50.5kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290234(CHEMBL440692 | N-[2-(2-Hydroxy-7-methoxy-naphthale...)
Affinity DataKi:  2.20nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9691(SCH446211 (SCH6) | TERT-BUTYL [(1S)-1-({(1R,2S,5S)...)
Affinity DataKi:  3.80nM ΔG°:  -48.9kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290239(CHEMBL78751 | N-{2-[2-(2-Hydroxy-ethoxy)-7-methoxy...)
Affinity DataKi:  4.30nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12493((2S)-({N-[3-({[(7R,9S,12S)-12-cyclohexyl-5,5-dimet...)
Affinity DataKi:  6nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187938(3-{(7R,9S,12S)-9-[1-((S)-dimethylcarbamoyl-phenyl-...)
Affinity DataKi:  6nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290237(CHEMBL82135 | N-[2-(2-Butoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12483((2S)-({N-[3-({[(5S,8S,10R)-5-cyclohexyl-3,6-dioxo-...)
Affinity DataKi:  7nM ΔG°:  -47.3kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290237(CHEMBL82135 | N-[2-(2-Butoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  7.70nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12287(SCH 491762 | tert-butyl N-[(1S)-2-[(1R,2S,5S)-2-[(...)
Affinity DataKi:  8nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12476((2S)-({N-[(3S)-3-({[(7R,9S,12S)-12-cyclohexyl-11,1...)
Affinity DataKi:  8nM ΔG°:  -47.0kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187936((7R,9S,12S)-12-cyclohexyl-11,14-dioxo-2,6-dioxa-10...)
Affinity DataKi:  8nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290241(CHEMBL311106 | N-[2-(7-Methoxy-2-propoxy-naphthale...)
Affinity DataKi:  8.10nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290236(CHEMBL80792 | N-{2-[2-(2-Dimethylamino-ethoxy)-7-m...)
Affinity DataKi:  10nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12475((2S)-({N-[3-({[(7R,9S,12S)-12-cyclohexyl-11,14-dio...)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9689(SCH446211 (SCH6) Analog 22 | tert-butyl N-[(2S)-1-...)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9686(2-methylpropyl N-[(1S)-1-cyclohexyl-2-[(1R,2S,5S)-...)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9684(2-methylpropyl N-[(2S)-1-[(3aR,4S,6aR)-4-({1-[({[(...)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12484((2S)-({N-[3-({[(7R,9S,12S)-12-cyclohexyl-11,14-dio...)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187934((7R,9S,12S)-12-cyclohexyl-19-methyl-11,14-dioxo-2,...)
Affinity DataKi:  12nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12309((1R,5S)-N-[3-amino-1-(cyclopropylmethyl)-2,3-dioxo...)
Affinity DataKi:  13nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12311((1R,5S)-N-[3-Amino-1-(cyclobutylmethyl)-2,3-dioxop...)
Affinity DataKi:  14nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9688(SCH446211 (SCH6) Analog 21 | tert-butyl N-[(2S)-1-...)
Affinity DataKi:  14nM ΔG°:  -45.6kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9685(2-methylpropyl N-[(2S)-1-[(1S,3aR,6aS)-1-({1-[({[(...)
Affinity DataKi:  15nM ΔG°:  -45.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12480((2S)-({N-[(3S)-3-({[(7R,9S,12S)-12-tert-butyl-11,1...)
Affinity DataKi:  15nM ΔG°:  -45.4kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12307((1R,5S)-N-[3-amino-1-(cyclobutylmethyl)-2,3-dioxop...)
Affinity DataKi:  16nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12492(Proline-Based Macrocycle 44 | tert-butyl (2S)-({N-...)
Affinity DataKi:  16nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290241(CHEMBL311106 | N-[2-(7-Methoxy-2-propoxy-naphthale...)
Affinity DataKi:  16nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9687(2-methylpropyl N-[(2S)-1-[(1R,2S,5S)-2-({1-[({[(S)...)
Affinity DataKi:  16nM ΔG°:  -45.2kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12494((2S)-({N-[3-({[(7R,9S,12S)-12-tert-butyl-5,5-dimet...)
Affinity DataKi:  17nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9683(2-methylpropyl N-[(2S)-1-[(2S,4R)-4-(tert-butoxy)-...)
Affinity DataKi:  19nM ΔG°:  -44.8kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187930(4-{(7R,9S,12S)-9-[1-((S)-dimethylcarbamoyl-phenyl-...)
Affinity DataKi:  19nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12495((2S)-({N-[3-({[(7R,9S,12S)-12-isopropyl-5,5-dimeth...)
Affinity DataKi:  19nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290235(CHEMBL78338 | {2-[7-Methoxy-1-(2-propionylamino-et...)
Affinity DataKi:  23nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM12286(1,1-Dimethylethyl-[1(S)-cyclohexyl-2-[(1R,5S)-2(S)...)
Affinity DataKi:  25nMAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187935((6R,8S,11S)-11-cyclohexyl-10,13-dioxo-2,5-dioxa-9,...)
Affinity DataKi:  25nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9679(2-methylpropyl N-[(1S)-1-cyclohexyl-2-[(3S)-3-({1-...)
Affinity DataKi:  26nM ΔG°:  -44.0kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50187929((7R,9S,12S)-12-cyclohexyl-15-methyl-11,14-dioxo-2,...)
Affinity DataKi:  26nMAssay Description:Binding affinity to HCV NS3 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9680(2-methylpropyl N-[(1S)-1-cyclohexyl-2-[(8S)-8-({1-...)
Affinity DataKi:  26nM ΔG°:  -44.0kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus (HCV genotype 1a, isolate H))
Schering-Plough Research Institute

LigandPNGBDBM9681(2-methylpropyl N-[(1S)-1-cyclohexyl-2-[(3S)-3-({1-...)
Affinity DataKi:  28nM ΔG°:  -43.8kJ/molepH: 6.5 T: 2°CAssay Description:Proteolytic cleavage of the ester linkage between the Nva (L-norvaline) and the chromophore (PAP) was monitored for change in absorbance at 370 nm. I...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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