Affinity DataKi: 0.0190nMAssay Description:Inhibition of human plasma kallikrein by Michaelis-menten analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate after 10 mins by UV/Vis photometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Inhibition of human plasmin using tosyl-Gly-Pro-Lys-pNA as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrateMore data for this Ligand-Target Pair
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Inhibition of activated protein kinase C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Inhibition of human plasmin using tosyl-Gly-Pro-Lys-pNA as substrate after 10 mins by UV/Vis photometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrate after 10 mins by UV/Vis photometryMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human plasmin using tosyl-Gly-Pro-Lys-pNA as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human plasmin using tosyl-Gly-Pro-Lys-pNA as substrate after 10 mins by UV/Vis photometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of human plasmin by Michaelis-menten analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of human plasmin using tosyl-Gly-Pro-Lys-pNA as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human plasmin assessed as reduction in proteolysis activity in presence of fibrinogen after 90 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of human plasmin assessed as reduction in proteolysis activity in presence of fibrinogen after 90 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Inhibition of human plasma kallikrein using S2302 as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of urokinase-type plasminogen activator (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Inhibition of urokinase-type plasminogen activator (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of plasmin (unknown origin)More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair