Compile Data Set for Download or QSAR
maximum 50k data
Found 29 with Last Name = 'placanica' and Initial = 'g'
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133069(3'-Ethylamino-[1,1';2',1'']terphenyl-4'-carbaldehy...)
Affinity DataKi:  0.0480nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133070(CHEMBL335465 | [1,1';2',1'']Terphenyl-4'-carbaldeh...)
Affinity DataKi:  0.150nMAssay Description:Relative binding affinity for human estrogen receptor alpha compared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133070(CHEMBL335465 | [1,1';2',1'']Terphenyl-4'-carbaldeh...)
Affinity DataKi:  0.270nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133069(3'-Ethylamino-[1,1';2',1'']terphenyl-4'-carbaldehy...)
Affinity DataKi:  0.470nMAssay Description:Relative binding affinity for human estrogen receptor alpha compared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133071(3'-Hydroxy-[1,1';2',1'']terphenyl-4'-carbaldehyde ...)
Affinity DataKi:  1.10nMAssay Description:Relative binding affinity for human estrogen receptor alpha compared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133071(3'-Hydroxy-[1,1';2',1'']terphenyl-4'-carbaldehyde ...)
Affinity DataKi:  1.70nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133072(3'-Amino-[1,1';2',1'']terphenyl-4'-carbaldehyde ox...)
Affinity DataKi:  2.20nMAssay Description:Relative binding affinity for human estrogen receptor alpha compared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133072(3'-Amino-[1,1';2',1'']terphenyl-4'-carbaldehyde ox...)
Affinity DataKi:  2.80nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133068(3'-Methylamino-[1,1';2',1'']terphenyl-4'-carbaldeh...)
Affinity DataKi:  3.70nMAssay Description:Relative binding affinity for human estrogen receptor alpha compared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50133068(3'-Methylamino-[1,1';2',1'']terphenyl-4'-carbaldeh...)
Affinity DataKi:  5.20nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  100nMAssay Description:Relative binding affinity for human estrogen receptor betacompared to [3H]-estradiolMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  100nMAssay Description:Binding affinity for human estrogen receptor alpha by displacement of [3H]-estradiolMore data for this Ligand-Target Pair
LigandPNGBDBM50051832(CHEMBL440280 | [((2E,6E,10E)-3,7,11,15-Tetramethyl...)
Affinity DataIC50:  66nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136457(CHEMBL136472 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50:  111nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136461(CHEMBL139238 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50:  146nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136459(CHEMBL139377 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50:  151nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136460(CHEMBL138033 | [((2E,6E,10E)-3,7,11,15-Tetramethyl...)
Affinity DataIC50:  275nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136458(CHEMBL134682 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50:  566nMAssay Description:In vitro inhibition of Geranylgeranyl protein transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50051832(CHEMBL440280 | [((2E,6E,10E)-3,7,11,15-Tetramethyl...)
Affinity DataIC50:  3.50E+3nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136460(CHEMBL138033 | [((2E,6E,10E)-3,7,11,15-Tetramethyl...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136458(CHEMBL134682 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136459(CHEMBL139377 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136457(CHEMBL136472 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50136461(CHEMBL139238 | [1-((2E,6E,10E)-3,7,11,15-Tetrameth...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of farnesyl protein transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity for human estrogen receptor alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.5nMAssay Description:Displacement of [3H]estradiol from human ERbetaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50192460(4-(4-hydroxyphenyl)-N-methyl-3-phenylanthranylaldo...)
Affinity DataKd:  3.70nMAssay Description:Displacement of [3H]estradiol from human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.200nMAssay Description:Displacement of [3H]estradiol from human ERalphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKd:  0.5nMAssay Description:Binding affinity for human estrogen receptor betaMore data for this Ligand-Target Pair