TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Concentration inhibiting Clostridium histolyticum collagenase.More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Technical University Of Denmark
Curated by ChEMBL
Technical University Of Denmark
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against Clostridium histolyticum CollagenaseMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 5.75E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 8.51E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 4.37E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 6.03E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 7.94E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 6.31E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 4.40E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 8.60E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 5.80E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 520nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 525nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 6.40E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 8.00E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: 6.00E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Uit The Arctic University Of Norway
Curated by ChEMBL
Uit The Arctic University Of Norway
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair