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Found 400 with Last Name = 'reboud-ravaux' and Initial = 'm'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430967(CHEMBL2337848)
Affinity DataKi:  2.30nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430968(CHEMBL2337847)
Affinity DataKi:  6nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430962(CHEMBL2337843)
Affinity DataKi:  10nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430969(CHEMBL2337846)
Affinity DataKi:  11nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)
Affinity DataKi:  11nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430970(CHEMBL2337845)
Affinity DataKi:  11nMAssay Description:Competitive inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universit£

Curated by ChEMBL
LigandPNGBDBM50485783(CHEMBL2164408)
Affinity DataKi:  50nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430963(CHEMBL2337842)
Affinity DataKi:  67nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156909(CHEMBL376817 | methyl (2S)-3-carbamoyl-2-[(2S)-2-[...)
Affinity DataKi:  80nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universit£

Curated by ChEMBL
LigandPNGBDBM50485784(CHEMBL2164407)
Affinity DataKi:  90nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  100nMAssay Description:Inhibition of dimerization of HIV1 protease 150V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430964(CHEMBL2337841)
Affinity DataKi:  101nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156906(CHEMBL375050 | methyl (2S)-2-[(2S)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  130nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universit£

Curated by ChEMBL
LigandPNGBDBM50485785(CHEMBL2164409)
Affinity DataKi:  150nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430963(CHEMBL2337842)
Affinity DataKi:  200nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191464(CHEMBL212749 | methyl (2S)-2-[(2S)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  200nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  200nMAssay Description:Inhibition of dimerization of HIV1 protease ANAM-11 mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156901((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  230nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  240nMAssay Description:Inhibition of dimerization of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156902((S)-methyl 2-((S)-2-((S)-2-(4-(2-(4-((2S,3S)-1-((2...)
Affinity DataKi:  250nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051763(2-iodophenyl 6-(chloromethyl)-2-oxo-2H-chromene-3-...)
Affinity DataKi:  250nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430964(CHEMBL2337841)
Affinity DataKi:  316nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM23563(3-Carboxylate-coumarin deriv., 3 | CHEMBL13357 | p...)
Affinity DataKi:  340nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051762(6-Chloromethyl-2-oxo-2H-chromene-3-carboxylic acid...)
Affinity DataKi:  380nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135844((2S,8S)-2-[({[({[(1S)-1-{[(1S,2R)-2-(benzyloxy)-1-...)
Affinity DataKi:  400nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156903((S)-methyl 2-((2S,3R)-3-hydroxy-2-((2S,3S)-2-(4-(7...)
Affinity DataKi:  400nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156910((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  410nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156908((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  420nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease D30N mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease G48V/L90M mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156904((S)-tert-butyl 5-((S)-1-amino-4-methyl-1-oxopentan...)
Affinity DataKi:  530nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universit£

Curated by ChEMBL
LigandPNGBDBM50074687(2-[2-(2-{4-[7-(3-{1-[1-(1-Methoxycarbonyl-2-methyl...)
Affinity DataKi:  560nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50074687(2-[2-(2-{4-[7-(3-{1-[1-(1-Methoxycarbonyl-2-methyl...)
Affinity DataKi:  560nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universit£

Curated by ChEMBL
LigandPNGBDBM50485786(CHEMBL2164074)
Affinity DataKi:  700nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Université

Curated by ChEMBL
LigandPNGBDBM50051761(2-chlorophenyl 6-(chloromethyl)-2-oxo-2H-chromene-...)
Affinity DataKi:  790nMAssay Description:Compound was tested for the binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156911((S)-5-((S)-1-amino-4-methyl-1-oxopentan-2-ylamino)...)
Affinity DataKi:  900nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156905((S)-methyl 2-((2S,3R)-3-hydroxy-2-(4-(7-(4-((S)-1-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156914((S)-methyl 2-((S)-2-((S)-2-(4-(7-(4-((2S,3S)-1-((2...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156913((S)-methyl 2-((2S,3R)-3-hydroxy-2-(4-(7-(4-((S)-1-...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156912(CHEMBL376602 | methyl (2S)-2-[(2S,3R)-2-[(2S,3R)-3...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156907((S)-methyl 2-((S)-2-((S)-2-(4-(7-(4-((S)-5-amino-1...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataKi:  2.43E+3nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50156902((S)-methyl 2-((S)-2-((S)-2-(4-(2-(4-((2S,3S)-1-((2...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM32709((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-met...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of dimerization of HIV1 protease MDR-HM mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185622(Apam-YET | CHEMBL210325)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430966(CHEMBL2337849)
Affinity DataKi:  5.03E+3nMAssay Description:Mixed type inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135845(Bicyclic Guanidinium Subunit | CHEMBL266754)
Affinity DataKi:  5.25E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50135842(Bicyclic Guanidinium Subunit | CHEMBL386994)
Affinity DataKi:  6.00E+3nMAssay Description:Competitive inhibition against HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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