TargetSigma non-opioid intracellular receptor 1(RAT)
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat brain membranes by competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.780nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat brain membranes by competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat brain membranes by competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.850nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat brain membranes by competitive binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 0.910nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in rat brain membranes by competitive binding assayMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to emopamil binding proteinMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 13.9nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 404nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 3.66E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 5.21E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 5.57E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 7.55E+3nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-B in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
General Hospital Of Pla
Curated by ChEMBL
General Hospital Of Pla
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair