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Found 44 with Last Name = 'ren' and Initial = 'xd'
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382321(CHEMBL2024688)
Affinity DataIC50:  1nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382322(CHEMBL2024689)
Affinity DataIC50:  1nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382324(CHEMBL2024691)
Affinity DataIC50:  2nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382320(CHEMBL2024687)
Affinity DataIC50:  3nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382318(CHEMBL2024685)
Affinity DataIC50:  4nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382319(CHEMBL2024686)
Affinity DataIC50:  4nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382325(CHEMBL2024693)
Affinity DataIC50:  5nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382323(CHEMBL2024690)
Affinity DataIC50:  6nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382317(CHEMBL2024684)
Affinity DataIC50:  13nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382318(CHEMBL2024685)
Affinity DataIC50:  44nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382325(CHEMBL2024693)
Affinity DataIC50:  46nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382324(CHEMBL2024691)
Affinity DataIC50:  47nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivin receptor type-1B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382317(CHEMBL2024684)
Affinity DataIC50:  59nMAssay Description:Inhibition of ALK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382321(CHEMBL2024688)
Affinity DataIC50:  61nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382326(CHEMBL2024692)
Affinity DataIC50:  69nMAssay Description:Inhibition of ALK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382323(CHEMBL2024690)
Affinity DataIC50:  73nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382319(CHEMBL2024686)
Affinity DataIC50:  135nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382317(CHEMBL2024684)
Affinity DataIC50:  211nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382322(CHEMBL2024689)
Affinity DataIC50:  274nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382320(CHEMBL2024687)
Affinity DataIC50:  695nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382326(CHEMBL2024692)
Affinity DataIC50:  708nMAssay Description:Inhibition of ALK5 in mouse NIH/3T3 cells by smad binding element reporter based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172943(5-chloro-N'-(o-tolylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172934(5-chloro-N'-(m-tolylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172945(CHEMBL205902 | N'-(phenylsulfonyl)dibenzo[b,d]fura...)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172944(5-bromo-N'-(phenylsulfonyl)benzofuran-2-carbohydra...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172940(CHEMBL437702 | N'-[(3-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, mitochondrial(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172933(5-chloro-N'-(2-(trifluoromethyl)phenylsulfonyl)-1H...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rat BCATmMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172931(CHEMBL205475 | N'-[(2-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172942(5-chloro-N'-(phenylsulfonyl)benzofuran-2-carbohydr...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase receptor R3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50382317(CHEMBL2024684)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of ALK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172932(5-chloro-N'-(2-chlorophenylsulfonyl)-1H-indole-2-c...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172947(5-methoxy-N'-(phenylsulfonyl)benzofuran-2-carbohyd...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172930(CHEMBL379025 | N'-[(2-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172936(CHEMBL437697 | N'-(phenylsulfonyl)quinoline-6-carb...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172937(5-bromo-N'-(phenylsulfonyl)-1H-indole-2-carbohydra...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172929(CHEMBL205220 | N'-(phenylsulfonyl)benzofuran-2-car...)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172928(CHEMBL382232 | N'-(phenylsulfonyl)quinoline-3-carb...)
Affinity DataIC50:  3.33E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172941(CHEMBL205274 | N'-[(3-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50: >3.50E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172935(CHEMBL207686 | N'-(phenylsulfonyl)-1H-indole-2-car...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172946(CHEMBL205044 | N'-[(4-chlorophenyl)sulfonyl]dibenz...)
Affinity DataIC50:  3.72E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172938(CHEMBL380652 | N'-[(4-methylphenyl)sulfonyl]dibenz...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBranched-chain-amino-acid aminotransferase, cytosolic(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50172939(5-methoxy-N'-(phenylsulfonyl)-1H-indole-2-carbohyd...)
Affinity DataIC50:  5.68E+4nMAssay Description:Inhibition of human BCATcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed