Compile Data Set for Download or QSAR
maximum 50k data
Found 78 with Last Name = 'ronken' and Initial = 'e'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50403670(CHEMBL311015)
Affinity DataKi:  0.229nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50403668(CHEMBL312339)
Affinity DataKi:  0.288nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50039824(CHEMBL81728 | N-{2-[4-(2,3-Dihydro-benzo[1,4]dioxi...)
Affinity DataKi:  0.295nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50039818(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(4-phenyl-...)
Affinity DataKi:  0.324nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  0.501nMAssay Description:Compound was tested for inhibition constant against 5-hydroxytryptamine 1A receptor in rat frontal cortex membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50039814(4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin...)
Affinity DataKi:  0.676nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM85079(2-[4-[4-[(7-Chloro-2,3-dihydro-1,4-benzodioxin)-5-...)
Affinity DataKi:  0.708nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50216215(CHEMBL81095)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50216214(CHEMBL311976)
Affinity DataKi:  1.20nMAssay Description:Compound was tested for its potency against 5-hydroxytryptamine 1A receptor in rat frontal cortex membranes (experiment 2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50039811(4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin...)
Affinity DataKi:  1.30nMAssay Description:Compound was tested for its potency against 5-hydroxytryptamine 1A receptor in rat frontal cortex membranes (experiment 1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50454759(Flesinoxan)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50005127(1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-b...)
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50230537((S)-3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)...)
Affinity DataKi:  7.80nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138899(3-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  13.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138902(CHEMBL160767 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  16.1nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138903(CHEMBL350924 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  16.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138897(CHEMBL351123 | Naphthalene-2-sulfonic acid 1-[3-(4...)
Affinity DataKi:  21.8nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138921(CHEMBL158138 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  22.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138912(CHEMBL156556 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  24.2nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM29094((+/-)-SLV319 | (S)-3-(4-chlorophenyl)-N-(4-chlorop...)
Affinity DataKi:  25nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50216216(CHEMBL81733)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138915(CHEMBL156264 | N-[1-[(S)-3-(4-Chloro-phenyl)-4-phe...)
Affinity DataKi:  35.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138900(CHEMBL157591 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  36.5nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138919(CHEMBL158502 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  52.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138918(CHEMBL348174 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  54.2nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138923(4-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  70.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138909(2-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  75.4nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138901(CHEMBL349771 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  119nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138911(CHEMBL158779 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  170nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138904(CHEMBL158610 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  196nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138895(CHEMBL158935 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  197nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138916(4-Chloro-N-[1-[3-(4-fluoro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  214nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138907(CHEMBL345466 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  221nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138910(CHEMBL158837 | N-[1-[3,4-Bis-(4-chloro-phenyl)-4,5...)
Affinity DataKi:  255nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138906(4-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  280nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138896(CHEMBL157149 | N-[1-[(R)-3-(4-Chloro-phenyl)-4-phe...)
Affinity DataKi:  293nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138908(CHEMBL347454 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  338nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138905(4-Chloro-N-[1-[3-(4-chloro-phenyl)-4-(4-fluoro-phe...)
Affinity DataKi:  584nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138917(CHEMBL348299 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  713nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138913(4-Chloro-N-[1-[(R)-3-(4-chloro-phenyl)-4-phenyl-4,...)
Affinity DataKi:  894nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138912(CHEMBL156556 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138913(4-Chloro-N-[1-[(R)-3-(4-chloro-phenyl)-4-phenyl-4,...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138900(CHEMBL157591 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138909(2-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138898(CHEMBL155752 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138908(CHEMBL347454 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138902(CHEMBL160767 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138899(3-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138898(CHEMBL155752 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Affinity to displace CP-55,940 binding from Cannabinoid receptor 2 of human expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 78 total ) | Next | Last >>
Jump to: