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Found 654 with Last Name = 'salunke' and Initial = 'db'
TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406601(CHEMBL5276854)
Affinity DataKi:  16nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
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TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406600(CHEMBL5267159)
Affinity DataKi:  22nMAssay Description:Negative log concentration of antagonist was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608747(CHEMBL5271653)
Affinity DataKi:  25nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608741(CHEMBL5284391)
Affinity DataKi:  41nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608748(CHEMBL5287590)
Affinity DataKi:  86nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406599(CHEMBL5276410)
Affinity DataKi:  91nMAssay Description:Negative log concentration of antagonistic compound was determined on 5-hydroxytryptamine 2B receptor of Rat stomach fundusMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608744(CHEMBL270735)
Affinity DataKi:  120nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608743(CHEMBL5280544)
Affinity DataKi:  140nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608742(CHEMBL5276994)
Affinity DataKi:  210nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50183456(CHEMBL425403 | N-methyl-N'-9-phenanthrylimidodicar...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50184688(CHEMBL377236 | Caulerpin)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421815(CHEMBL5276478)
Affinity DataKi:  2.55E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421812(CHEMBL5279244)
Affinity DataKi:  4.21E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421811(CHEMBL5287944)
Affinity DataKi:  5.38E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421811(CHEMBL5287944)
Affinity DataKi:  6.45E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608746(CHEMBL5275669)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPDB
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TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421815(CHEMBL5276478)
Affinity DataKi:  8.39E+3nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421813(CHEMBL5272039)
Affinity DataKi:  9.29E+3nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetSodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421814(CHEMBL5287717)
Affinity DataKi:  1.18E+4nMAssay Description:Binding affinity to NTCP (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421814(CHEMBL5287717)
Affinity DataKi:  1.52E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421813(CHEMBL5272039)
Affinity DataKi:  1.56E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIleal sodium/bile acid cotransporter(Homo sapiens (Human))TBA
LigandPNGBDBM50421812(CHEMBL5279244)
Affinity DataKi:  2.04E+4nMAssay Description:Binding affinity to ASBT (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50428658(MITOMYCIN | Mitomycin C | Mitosol | Mitozytrex | M...)
Affinity DataKi:  2.50E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608745(CHEMBL5272397)
Affinity DataKi:  7.00E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  9.40E+4nMAssay Description:Binding affinity to human recombinant IDO1 assessed as inhibition constant using L-tryptophan as substrate incubated for 10 mins by methylene blue dy...More data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM24813(Brassinin, 1 | N-(1H-indol-3-ylmethyl)(methylsulfa...)
Affinity DataKi:  9.77E+4nMAssay Description:Binding affinity to IDO1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50562506(CHEMBL4791168)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of IDO1 in human HeLa cells using L-tryptophan as substrate incubated for 48 hrs by absorbance based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50590774(CHEMBL5203175)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of IDO1 in human HeLa cells assessed as inhibition of kynurenine production incubated for 30 mins by microplate reader based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608773(CHEMBL5265978)
Affinity DataIC50:  28nMAssay Description:Inhibition of IDO1 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608773(CHEMBL5265978)
Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant N-terminal his6-tagged IDO1 expressed in Escherichia coli BL21 using L-tryptophan as substrate incubated for 1 hr by ...More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50084419(Andrographolide | CHEBI:65408)
Affinity DataIC50:  56nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608750(CHEMBL5275082)
Affinity DataIC50:  71nMAssay Description:Inhibition of human recombinant IDO1 using L-tryptophan as substrate incubated for 10 mins by absorbance based analysisMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608773(CHEMBL5265978)
Affinity DataIC50:  92nMAssay Description:Inhibition of human recombinant N-terminal his6-tagged IDO1 expressed in Escherichia coli BL21 using L-tryptophan as substrate incubated for 1 hr by ...More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50562506(CHEMBL4791168)
Affinity DataIC50:  94nMAssay Description:Inhibition of human N-terminal his-tagged IDO1 expressed in Escherichia coli using L-tryptophan as substrate by UV absorption based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608775(CHEMBL5287332)
Affinity DataIC50:  100nMAssay Description:Inhibition of IDO1 in human HeLa cells assessed as inhibition of kynurenine production incubated for 30 mins by microplate reader based analysisMore data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608772(CHEMBL5271416)
Affinity DataIC50:  100nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50562515(CHEMBL4740878)
Affinity DataIC50:  130nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetIndoleamine 2,3-dioxygenase 1(Mus musculus)TBA
LigandPNGBDBM50608761(CHEMBL4534417)
Affinity DataIC50:  160nMAssay Description:Inhibition of mouse IDO1 using L-tryptophan as substrate by methylene blue dye based analysisMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608765(CHEMBL5288553)
Affinity DataIC50:  199nMAssay Description:Inhibition of human IDO1More data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM387356(N3-(3-Chloro- 4-fluorophenyl) furo[2,3- c]pyridine...)
Affinity DataIC50: <200nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500136(CHEMBL3746040)
Affinity DataIC50:  240nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608738(CHEMBL5283627)
Affinity DataIC50:  270nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608740(CHEMBL3765916)
Affinity DataIC50:  300nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608766(CHEMBL5281451)
Affinity DataIC50:  331nMAssay Description:Inhibition of human recombinant IDO1 using L-tryptophan as substrate incubated for 45 mins by methylene blue dye based microplate reader analysisMore data for this Ligand-Target Pair
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TargetToll-like receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50406601(CHEMBL5276854)
Affinity DataIC50:  361nMAssay Description:Antagonistic activity against Bradykinin receptor B1 of rat ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608739(CHEMBL5285306)
Affinity DataIC50:  400nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM81348(β-Lapachone (A3) | Beta lapachone | R115 (Rea...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human recombinant IDO1 expressed in Escherichia coliMore data for this Ligand-Target Pair
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608729(CHEMBL5276255)
Affinity DataIC50:  500nMAssay Description:Inhibition of IDO1 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608768(CHEMBL4542547)
Affinity DataIC50:  500nMAssay Description:Inhibition of human IDO1 expressed in Escherichia coli using L-tryptophan as substrate incubated for 30 mins by methylene blue dye based microplate r...More data for this Ligand-Target Pair
Ligand Info
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TargetIndoleamine 2,3-dioxygenase 1(Mus musculus)TBA
LigandPNGBDBM50608759(CHEMBL5267145)
Affinity DataIC50:  510nMAssay Description:Inhibition of mouse IDO1 using L-tryptophan as substrate by methylene blue dye based analysisMore data for this Ligand-Target Pair
Ligand Info
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