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Found 408 with Last Name = 'santana' and Initial = 'l'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073274(3-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  0.790nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073273(3,4-Dimethyl-7-[3-(4-phenyl-piperazin-1-yl)-propox...)
Affinity DataKi:  5.30nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073272(4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  5.5nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073271(7-[3-(4-Phenyl-piperazin-1-yl)-propoxy]-chromen-2-...)
Affinity DataKi:  5.60nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073273(3,4-Dimethyl-7-[3-(4-phenyl-piperazin-1-yl)-propox...)
Affinity DataKi:  5.90nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50409503(CHEMBL310153)
Affinity DataKi:  6.5nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073274(3-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  11nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404053(CHEMBL51767)
Affinity DataKi:  12nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073272(4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  14nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073271(7-[3-(4-Phenyl-piperazin-1-yl)-propoxy]-chromen-2-...)
Affinity DataKi:  16nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404050(CHEMBL298108)
Affinity DataKi:  18nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073274(3-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  19nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50409510(CHEMBL308480)
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50409493(CHEMBL310734)
Affinity DataKi:  25nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073273(3,4-Dimethyl-7-[3-(4-phenyl-piperazin-1-yl)-propox...)
Affinity DataKi:  45nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50073272(4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  46nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404047(CHEMBL52384)
Affinity DataKi:  48nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073271(7-[3-(4-Phenyl-piperazin-1-yl)-propoxy]-chromen-2-...)
Affinity DataKi:  50nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  52nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Vigo

Curated by ChEMBL
LigandPNGBDBM50073272(4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  74nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50453056(CHEMBL73675)
Affinity DataKi:  74nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50453055(CHEMBL72649)
Affinity DataKi:  78nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]spiperone binding to the dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404052(CHEMBL51681)
Affinity DataKi:  81nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  98nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the Dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404049(CHEMBL48205)
Affinity DataKi:  129nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404047(CHEMBL52384)
Affinity DataKi:  138nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404053(CHEMBL51767)
Affinity DataKi:  174nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50519753(CHEMBL4526845)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404051(CHEMBL265805)
Affinity DataKi:  324nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409510(CHEMBL308480)
Affinity DataKi:  324nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409493(CHEMBL310734)
Affinity DataKi:  380nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404049(CHEMBL48205)
Affinity DataKi:  537nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404048(CHEMBL48194)
Affinity DataKi:  562nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50453056(CHEMBL73675)
Affinity DataKi:  741nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50453055(CHEMBL72649)
Affinity DataKi:  912nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50073272(4-Methyl-7-[3-(4-phenyl-piperazin-1-yl)-propoxy]-c...)
Affinity DataKi:  933nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404052(CHEMBL51681)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409503(CHEMBL310153)
Affinity DataKi:  1.35E+3nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM82053(8-(2-Furyl)theophylline | US9138393, Theophylline ...)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]NECA from human adenosine receptor A2A expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404048(CHEMBL48194)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404051(CHEMBL265805)
Affinity DataKi:  2.34E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50519760(CHEMBL3950921)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago

Curated by ChEMBL
LigandPNGBDBM50404050(CHEMBL298108)
Affinity DataKi:  3.09E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM95955(MLS000693557 | N-(2-ketochromen-3-yl)benzamide | N...)
Affinity DataKi:  3.24E+3nMAssay Description:The radioligands used were 1 nM (2R,3R,4S,5R)-2-(2-chloro-6-cyclopentylamino-purin-9-yl)-5-hydroxymethyl-tetrahydro-3,4-diol ([3H]CCPA) for hA1, 10 n...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50519760(CHEMBL3950921)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50519762(CHEMBL4565447)
Affinity DataKi:  3.93E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50344059(8-Hydroxy-3-phenylcoumarin | CHEMBL1777846)
Affinity DataKi:  4.62E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Porto

Curated by ChEMBL
LigandPNGBDBM50519754(CHEMBL1417172)
Affinity DataKi:  5.06E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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