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Found 331 with Last Name = 'savage' and Initial = 'm'
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513934(CHEMBL4443587)
Affinity DataKi:  0.360nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513931(CHEMBL4444446)
Affinity DataKi:  0.530nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205423(US9243020, 17 | US9815861, Example 17)
Affinity DataKi:  0.550nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001092(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  0.900nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50000335(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  1.80nMAssay Description:In Vitro evaluation for the binding affinity in homogenates of rat brain at Opioid receptor delta 1 by displacing [3H]- DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli assessed as inhibitory constant using 4-MUGlcNAc as substrate incubated for 20 mins...More data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205425(US9243020, 20 | US9815861, Example 20)
Affinity DataKi:  2.40nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001090(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  2.5nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM141965(US8927507, 16)
Affinity DataKi:  2.80nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205422(US9243020, 9 | US9815861, Example 9)
Affinity DataKi:  3nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513947(CHEMBL4545886)
Affinity DataKi:  3.30nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513960(CHEMBL4561925)
Affinity DataKi:  5.30nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513955(CHEMBL4483089)
Affinity DataKi:  5.5nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513957(CHEMBL4456515)
Affinity DataKi:  5.60nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001088((DPDPE)13-[2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  7nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205424(US9243020, 19 | US9815861, Example 19)
Affinity DataKi:  7.90nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513958(CHEMBL4473252)
Affinity DataKi:  9nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513939(CHEMBL4516713)
Affinity DataKi:  9.40nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001090(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  9.5nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205421(US9243020, 4 | US9815861, Example 4)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM142083(US8933040, 7)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513951(CHEMBL4583010)
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513940(CHEMBL4586062)
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  18nMAssay Description:In Vitro evaluation for the binding affinity in homogenates of rat brain at Opioid receptor delta 1 by displacing [3H]- DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513930(CHEMBL4543991)
Affinity DataKi:  20nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001093(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  21nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205428(US9243020, 33 | US9815861, Example 33)
Affinity DataKi:  23nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513944(CHEMBL4453820)
Affinity DataKi:  26nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205426(US9243020, 27 | US9815861, Example 27)
Affinity DataKi:  28nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513956(CHEMBL4448352)
Affinity DataKi:  29nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  32nMAssay Description:Dissociation rate constant of compound for mutant T46S Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  32nMAssay Description:Compound was evaluated for its binding affinity by displacement of [3H]- DAMPGO from opioid receptor mu by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513949(CHEMBL4476839)
Affinity DataKi:  35nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513952(CHEMBL4576476)
Affinity DataKi:  41nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205420(US9243020, 2 | US9815861, Example 2)
Affinity DataKi:  44nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001089(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  45nMAssay Description:Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513959(CHEMBL4465511)
Affinity DataKi:  50nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513950(CHEMBL4454814)
Affinity DataKi:  50nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513942(CHEMBL4436228)
Affinity DataKi:  58nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50000335(13-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-prop...)
Affinity DataKi:  58nMAssay Description:In Vitro evaluation for the binding affinity in homogenates of rat brain at opioid receptor mu by displacing [3H]- DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM205419(US9243020, 1 | US9815861, Example 1)
Affinity DataKi:  69nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513954(CHEMBL4527453)
Affinity DataKi:  70nMAssay Description:Inhibition of human OGA assessed as inhibitory constant using 4-methylumbelliferyl 2-acetamido-2-deoxy-beta-D-glucopyranoside as substrate incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513954(CHEMBL4527453)
Affinity DataKi:  70nMAssay Description:Inhibition of human beta hexosaminidase assessed as inhibitory constant using 4-methylumbelliferyl 2-acetamido-2-deoxy-beta-D-glucopyranoside as subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50513932(CHEMBL4541985)
Affinity DataKi:  72nMAssay Description:Inhibition of recombinant human OGAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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