TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant HER2 (675 to 1255) (unknown origin) expressed in baculovirus infected Sf9 insect cells using poly-Glu-Tyr as substrate incu...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 10.8nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 209nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 214nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 247nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 263nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 314nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 325nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 439nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 534nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 537nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 632nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 662nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 671nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 719nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 805nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 811nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 855nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His-tagged cytoplasmic c-MET kinase domain (956 to 1390 residues) phosphorylation expressed in baculovirus...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair