Compile Data Set for Download or QSAR
maximum 50k data
Found 132 with Last Name = 'sayed' and Initial = 'ka'
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50559346(CHEMBL4763836)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50559344(CHEMBL4796265)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332525(CHEMBL1630488 | N-(4-methoxyphenyl)-5-(4-nitrophen...)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50559342(CHEMBL4793731)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50559343(CHEMBL4783947)
Affinity DataIC50:  10nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM31340(2-methoxy-N-[(E)-3-[4-[3-methyl-4-(6-methylpyridin...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant HER2 (675 to 1255) (unknown origin) expressed in baculovirus infected Sf9 insect cells using poly-Glu-Tyr as substrate incu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332529(4-(9H-purin-6-ylamino)-2-((bis(2-chloroethyl)amino...)
Affinity DataIC50:  10.8nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50559345(CHEMBL4782561)
Affinity DataIC50:  12nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332538(CHEMBL1630452 | N-(3-chloro-4-methylphenyl)-5-(4-n...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332524(4-(5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)b...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332519(CHEMBL1630483 | N-(4-Methoxyphenyl)-5-(4-(trifluor...)
Affinity DataIC50:  53nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50161957(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(p...)
Affinity DataIC50:  60nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM50161957(4-Dimethylamino-but-2-enoic acid {4-[3-chloro-4-(p...)
Affinity DataIC50:  90nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Texas A&M University

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  96nMAssay Description:Inhibition of HER2 (unknown origin) in presence of substrate incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332534(2-(4-amino-5-(4-hydroxy-3-methoxyphenyl)pyrido[2,3...)
Affinity DataIC50:  113nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332540((Z)-5-(2,3-methylenedioxyphenyl)imidazolidine-2,4-...)
Affinity DataIC50:  138nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332503(5-(4-nitrophenyl)-N-phenyl-1,3,4-oxadiazol-2-amine...)
Affinity DataIC50:  209nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332532((E)-5-(3,4,5-trimethoxybenzylidene)imidazolidine-2...)
Affinity DataIC50:  214nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332502(4-(5-(phenylamino)-1,3,4-oxadiazol-2-yl)benzonitri...)
Affinity DataIC50:  247nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332533((Z)-3,3'-(4-((4-oxo-2-thioxothiazolidin-5-ylidene)...)
Affinity DataIC50:  263nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332522(CHEMBL1630486 | N-(4-Methoxyphenyl)-5-(4-(methylsu...)
Affinity DataIC50:  314nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332537(6-(4-fluorophenyl)-3-hydroxy-4-(4-methoxyphenyl)py...)
Affinity DataIC50:  325nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332500(5-(4-(Methylsulfonyl)phenyl)-N-phenyl-1,3,4-oxadia...)
Affinity DataIC50:  439nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332518(5-(4-Chlorophenyl)-N-(4-methoxyphenyl)-1,3,4-oxadi...)
Affinity DataIC50:  534nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332535((Z)-2-methoxy-5-((4-oxo-2-thioxothiazolidin-5-ylid...)
Affinity DataIC50:  537nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332498(5-(4-(Trifluoromethyl)phenyl)-N-phenyl-1,3,4-oxadi...)
Affinity DataIC50:  632nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332526(CHEMBL1630489 | N,5-Bis(4-methoxyphenyl)-1,3,4-oxa...)
Affinity DataIC50:  662nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332511(CHEMBL1630475 | N-(4-Chlorophenyl)-5-(4-(methylsul...)
Affinity DataIC50:  671nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332527(CHEMBL1630490 | N,5-bis(4-nitrophenyl)-1,3,4-oxadi...)
Affinity DataIC50:  710nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332513(4-(5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-ylamino)be...)
Affinity DataIC50:  719nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332520(CHEMBL1630484 | N-(4-Methoxyphenyl)-5-p-tolyl-1,3,...)
Affinity DataIC50:  805nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332514(CHEMBL1630478 | N-(4-Chlorophenyl)-5-(4-nitropheny...)
Affinity DataIC50:  811nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332510(CHEMBL1630474 | N-(4-Chlorophenyl)-5-(4-(methylmer...)
Affinity DataIC50:  855nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332496(CHEMBL1630460 | N,5-diphenyl-1,3,4-oxadiazol-2-ami...)
Affinity DataIC50:  980nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332515(CHEMBL1630479 | N-(4-chlorophenyl)-5-(4-methoxyphe...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332512(CHEMBL1630476 | N-(4-Chlorophenyl)-5-(4-(dimethyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332509(CHEMBL1630473 | N-(4-Chlorophenyl)-5-p-tolyl-1,3,4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332508(CHEMBL1630472 | N-(4-Chlorophenyl)-5-(4-(trifluoro...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332507(CHEMBL1630471 | N,5-Bis(4-chlorophenyl)-1,3,4-oxad...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332506(CHEMBL1630470 | N-(4-chlorophenyl)-5-phenyl-1,3,4-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332505(4-(5-(phenylamino)-1,3,4-oxadiazol-2-yl)phenol | C...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332504(5-(4-methoxyphenyl)-N-phenyl-1,3,4-oxadiazol-2-ami...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332501(5-(4-(dimethylamino)phenyl)-N-phenyl-1,3,4-oxadiaz...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332523(5-(4-(Dimethylamino)phenyl)-N-(4-methoxyphenyl)-1,...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332517(CHEMBL1630481 | N-(4-methoxyphenyl)-5-phenyl-1,3,4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332521(CHEMBL1630485 | N-(4-Methoxyphenyl)-5-(4-(methylth...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332516(4-(5-(4-chlorophenylamino)-1,3,4-oxadiazol-2-yl)ph...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50185608(CHEMBL3822800)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His-tagged cytoplasmic c-MET kinase domain (956 to 1390 residues) phosphorylation expressed in baculovirus...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM50332497(5-(4-chlorophenyl)-N-phenyl-1,3,4-oxadiazol-2-amin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
University Of Louisiana At Monroe

Curated by ChEMBL
LigandPNGBDBM38948(5-(4-methylphenyl)-N-phenyl-1,3,4-oxadiazol-2-amin...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant GSK3beta Z'-LYTE kinase assay kit methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 132 total ) | Next | Last >>
Jump to: