Compile Data Set for Download or QSAR
maximum 50k data
Found 95 with Last Name = 'sayre' and Initial = 'lm'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  3.60nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021495(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021493(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021499(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021498(1N,4N-di[4-cyclopropylmethyl-10,17-dihydroxy-(13R,...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  16nMAssay Description:The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  27nMAssay Description:Compound was tested for binding affinity against delta opioid receptor in guinea pig brain membrane using [3H]-EK as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021500(1N-[4-cyclopropylmethyl-10,17-dihydroxy-(13R,14R,1...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM224024(BDBM50241435 | Dynorphin A (1-13) | YGGFLRRXRPKLK)
Affinity DataKi:  50nMAssay Description:The compound was tested for binding activity towards opioid receptor mu in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021490(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-naloxone from Opioid receptor mu 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021492(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021501(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021497(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021502(1N,4N-di[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021504(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021491(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-EK from Opioid receptor delta 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021496(1N,4N-di[10,17-dihydroxy-4-methyl-(13S,14R,17R)-12...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50009674(4-Amino-N-[2-(4-amino-butyrylamino)-ethyl]-N-[2-((...)
Affinity DataKi:  3.73E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021494(1N-[10,17-dihydroxy-4-methyl-(13R,14R,17S)-12-oxa-...)
Affinity DataKi:  4.40E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50009677(4-Amino-N-[3-(4-amino-butyrylamino)-propyl]-N-{3-[...)
Affinity DataKi:  5.51E+3nMAssay Description:The compound was tested for binding activity towards opioid receptor kappa in guinea pig brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50021503(1N-[10,17-dihydroxy-4-methyl-(13R,14S,17S)-12-oxa-...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H]-DADLE from Opioid receptor kappa 1 in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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