Affinity DataKi: 0.0140nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity towards human estrogen receptor beta in a competitive binding assay using fluorescently labelled estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity towards human estrogen receptor alpha in a competitive binding assay using fluorescently labelled estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 184nMAssay Description:Antagonistic activity against estrogen receptor alpha in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataKi: 421nMAssay Description:Antagonistic activity against estrogen receptor beta in presence of 0.1 nM estradiolMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15.5nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataIC50: 165nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Half-maximum activation of human Thyroid hormone receptor beta 1 (hTRbeta1)More data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Half-maximum activation of human Thyroid hormone receptor beta 1 (hTRbeta1)More data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:Half-maximum activation of human Thyroid hormone receptor alpha1 (hTRalpha1)More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataIC50: >2.00E+3nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco
Curated by ChEMBL
University Of California San Francisco
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair