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maximum 50k data
Found 656 with Last Name = 'schrag' and Initial = 'm'
LigandPNGBDBM50343209(CHEMBL1773731 | N-(6-(6-Chloro-5-(3-chlorophenylsu...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343206(CHEMBL1773728 | N-(6-(6-Chloro-5-(3-(trifluorometh...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343203(CHEMBL1773604 | N-(6-(6-Chloro-5-(4-methoxyphenyls...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343210(CHEMBL1773732 | N-(6-(6-Chloro-5-(4-chlorophenylsu...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343211(CHEMBL1773733 | N-(6-(5-(3-tert-Butylphenylsulfona...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343207(CHEMBL1773729 | N-(6-(6-Chloro-5-(4-(trifluorometh...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343208(CHEMBL1773730 | N-(6-(6-Chloro-5-(2-chlorophenylsu...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343213(CHEMBL1773735 | N-(6-(6-Chloro-5-(2-fluorophenylsu...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343212(CHEMBL1773734 | N-(6-(6-Chloro-5-(4-tert-butylphen...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343205(CHEMBL1773606 | N-(6-(6-Chloro-5-(2-(trifluorometh...)
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343214(CHEMBL1773736 | N-(6-(6-Chloro-5-(3-fluorophenylsu...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343202(CHEMBL1773603 | N-(6-(5-(4-Methoxyphenylsulfonamid...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kdelta expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343204(CHEMBL1773605 | N-(6-(6-Chloro-5-(phenylsulfonamid...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343201(CHEMBL1773602 | N-(6-(6-Cyano-5-(4-methoxyphenylsu...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343197(CHEMBL1773599 | N-(6-(5-(4-Methoxyphenylsulfonamid...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)
Affinity DataKi:  2nMAssay Description:Inhibition of human PI3Kbeta expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of human PI3Kgamma expressed in Sf9 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50343198(CHEMBL1773600 | N-(6-(6-(4-Methoxyphenylsulfonamid...)
Affinity DataKi:  9nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343196(CHEMBL1773558 | N-(6-(2-(4-Methoxyphenylsulfonamid...)
Affinity DataKi:  13nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343232(CHEMBL1773559 | N-(6-(2-(4-Methoxyphenylthio)pyrim...)
Affinity DataKi:  18nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343235(CHEMBL1773077 | N-(6-(2-(3-Methoxybenzyloxy)pyrimi...)
Affinity DataKi:  18nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343246(CHEMBL1773572 | N-(6-(2-(2-Phenylpropan-2-ylamino)...)
Affinity DataKi:  24nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343225(CHEMBL1773592 | N-(6-(2-(3-Fluorophenylthio)pyrimi...)
Affinity DataKi:  31nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343227(CHEMBL1773594 | N-(6-(2-(2-Methylphenylthio)pyrimi...)
Affinity DataKi:  31nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)
Affinity DataKi:  31nMAssay Description:Inhibition of human VPS34 after 30 mins by fluorescence-based immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343242(CHEMBL1773568 | N-(6-(2-(3-Phenylpropoxy)pyrimidin...)
Affinity DataKi:  32nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343195(CHEMBL1773582 | N-(6-(2-(4-Methyl-N-methylphenylsu...)
Affinity DataKi:  38nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343216(CHEMBL1773583 | N-(6-(2-(Phenylthio)pyrimidin-4-yl...)
Affinity DataKi:  40nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343190(CHEMBL1773577 | N-(6-(2-(2-Fluorophenylsulfonamido...)
Affinity DataKi:  41nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343226(CHEMBL1773593 | N-(6-(2-(4-Fluorophenylthio)pyrimi...)
Affinity DataKi:  44nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343224(CHEMBL1773591 | N-(6-(2-(2-Fluorophenylthio)pyrimi...)
Affinity DataKi:  46nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343234(CHEMBL1773561 | N-(6-(2-(3-Methylbenzyloxy)pyrimid...)
Affinity DataKi:  47nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343217(CHEMBL1773584 | N-(6-(2-(Benzylthio)pyrimidin-4-yl...)
Affinity DataKi:  47nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343231(CHEMBL1773598 | N-(6-(2-(3-Methoxyphenylthio)pyrim...)
Affinity DataKi:  48nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343199(CHEMBL1773601 | N-(6-(3-(4-Methoxyphenylsulfonamid...)
Affinity DataKi:  48nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343215(CHEMBL1615188 | N-(6-(2-(methylthio)pyrimidin-4-yl...)
Affinity DataKi:  53nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343215(CHEMBL1615188 | N-(6-(2-(methylthio)pyrimidin-4-yl...)
Affinity DataKi:  53nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343228(CHEMBL1773595 | N-(6-(2-(3-Methylphenylthio)pyrimi...)
Affinity DataKi:  53nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343237(CHEMBL1773563 | N-(6-(2-(4-Methylbenzyloxy)pyrimid...)
Affinity DataKi:  58nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343238(CHEMBL1773564 | N-(6-(2-(4-Methoxybenzyloxy)pyrimi...)
Affinity DataKi:  58nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343229(CHEMBL1773596 | N-(6-(2-(4-Methylphenylthio)pyrimi...)
Affinity DataKi:  59nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343233(CHEMBL1773560 | N-(6-(2-(3-Fluorobenzyloxy)pyrimid...)
Affinity DataKi:  61nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343189(CHEMBL1773576 | N-(6-(2-(N-Ethyl-4-methoxyphenylsu...)
Affinity DataKi:  62nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343191(CHEMBL1773578 | N-(6-(2-(2-Fluoro-N-methylphenylsu...)
Affinity DataKi:  65nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343249(CHEMBL1773575 | N-(6-(2-(4-Methoxy-N-methylphenyls...)
Affinity DataKi:  76nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343194(CHEMBL1773581 | N-(6-(2-(4-Methylphenylsulfonamido...)
Affinity DataKi:  82nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343192(CHEMBL1773579 | N-(6-(2-(3-Fluorophenylsulfonamido...)
Affinity DataKi:  84nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50343221(CHEMBL1773588 | N-(6-(2-(Benzylamino)pyrimidin-4-y...)
Affinity DataKi:  85nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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