TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 0.00190nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCG by dilution assayMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 0.0521nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of ECG by dilution assayMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 0.109nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGC by dilution assayMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 0.281nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of quercetin by dilution assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand co-expressed with delta and kappa opioid receptor...More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand co-expressed with delta and kappa opioid receptor...More data for this Ligand-Target Pair
Affinity DataKi: 0.676nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 0.798nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of butein by dilution assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.891nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCGMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand singly expressed with delta or kappa receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.13nMAssay Description:Effect on binding to wild-type opioid receptor kappa 1 using [3H]diprenorphine in transiently expressed rat HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15nMAssay Description:Binding affinity towards rat opioid receptor kappa 1 was determined using [3H]diprenorphine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand co-expressed with delta and kappa opioid receptor...More data for this Ligand-Target Pair
Affinity DataKi: 1.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.19nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.24nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Binding affinity towards mouse delta-opioid receptor was determined using [3H]diprenorphine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.82nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.95nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand singly expressed with delta or kappa receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.63nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Inhibition of Plasmodium falciparum recombinant enoyl ACP reductase expressed in BL21 (DE3) cells with respect to crotonyl CoAMore data for this Ligand-Target Pair
Affinity DataKi: 4.27nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand co-expressed with delta and kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.62nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Compound was tested for binding affinity on intact HEK cells using [3H]diprenorphine as radioligand singly expressed with delta or kappa receptors.More data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 7.29nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of EGCGMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of ECGMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 8.25nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of EGCMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of quercetinMore data for this Ligand-Target Pair
Affinity DataKi: 12.3nMAssay Description:Effect on binding to kappa(Glu297Ala) opioid receptor, using [3H]diprenorphine in transiently expressed rat HEK293 cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 13.7nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of buteinMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
Affinity DataKi: 17.4nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 17.6nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
Affinity DataKi: 18.2nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20.3nMAssay Description:Binding affinity towards mouse delta-opioid receptor was determined using [3H]diprenorphine as radioligandMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of Plasmodium falciparum ENR in presence of triclosanMore data for this Ligand-Target Pair
Affinity DataKi: 27.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetEnoyl-acyl-carrier protein reductase(Plasmodium falciparum)
National Institute Of Immunology
Curated by ChEMBL
National Institute Of Immunology
Curated by ChEMBL
Affinity DataKi: 28.3nMAssay Description:Inhibition of Plasmodium falciparum ENR by fluorescence quenching in presence of ECGMore data for this Ligand-Target Pair
Affinity DataKi: 29.5nMAssay Description:Displacement of [125I]I-AB-MEAC from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair