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Found 103 with Last Name = 'shipway' and Initial = 'a'
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246998(CHEMBL505558 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246999(CHEMBL500474 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246997(CHEMBL505738 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  27nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246995(CHEMBL505048 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247004((3R,5S)-5-(((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-...)
Affinity DataKi:  29nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246992(CHEMBL498914 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246994(CHEMBL443101 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  41nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246996(CHEMBL506226 | {(R)-1-[(2S,4R)-2-[(S)-5-Amino-1-(b...)
Affinity DataKi:  45nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246991(CHEMBL509770 | benzyl (R)-1-((2S,3S)-2-(((S)-6-ami...)
Affinity DataKi:  49nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247002(((R)-1-{(2S,4R)-2-[(S)-5-Amino-1-(benzooxazole-2-c...)
Affinity DataKi:  60nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247000(CHEMBL446259 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  65nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247005((3R,5S)-5-(((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-...)
Affinity DataKi:  101nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247001(CHEMBL448873 | Phenyl-carbamic acid (3R,5S)-5-[(S)...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247003(CHEMBL501945 | {(R)-1-[(2S,4R)-2-[(S)-5-Amino-1-(b...)
Affinity DataKi:  176nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246990(CHEMBL454436 | benzyl (R)-1-((2S,3R)-2-(((S)-6-ami...)
Affinity DataKi:  267nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247006((3R,5S)-5-((S)-6-amino-1-(benzo[d]oxazol-2-yl)-1-o...)
Affinity DataKi:  510nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246993(CHEMBL507245 | benzyl (R)-1-((2S,4R)-2-(((S)-6-ami...)
Affinity DataKi:  1.04E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246989(CHEMBL501802 | benzyl (R)-1-((S)-2-(((S)-6-amino-1...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50247007(((R)-1-{(2S,4R)-2-[(S)-5-Amino-1-(benzooxazole-2-c...)
Affinity DataKi:  1.55E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246988(CHEMBL503925 | benzyl (S)-1-((S)-1-((S)-6-amino-1-...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246986(CHEMBL507205 | benzyl (S)-1-((S)-1-((S)-6-amino-1-...)
Affinity DataKi:  5.72E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246987(CHEMBL504394 | benzyl (S)-6-amino-1-((S)-1-((S)-6-...)
Affinity DataKi:  5.78E+3nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246985(CHEMBL507704 | benzyl (S)-6-amino-1-((S)-1-((S)-6-...)
Affinity DataKi:  1.52E+4nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246984(CHEMBL508055 | benzyl (S)-1-((S)-6-amino-1-(benzo[...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstasin(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50246983(CHEMBL509923 | benzyl (S)-1-((S)-6-amino-1-(benzo[...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human prostasinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380413(CHEMBL2018573)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380417(CHEMBL2018485)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380418(CHEMBL2018571)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380410(CHEMBL2018484)
Affinity DataIC50:  6.80nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380417(CHEMBL2018485)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380414(CHEMBL2018467)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380437(CHEMBL2018474)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380413(CHEMBL2018573)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380418(CHEMBL2018571)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380411(CHEMBL2018465)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380425(CHEMBL2018460)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380410(CHEMBL2018484)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380412(CHEMBL2018486)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380443(CHEMBL2018480)
Affinity DataIC50:  84nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380415(CHEMBL2018481)
Affinity DataIC50:  84.7nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380409(CHEMBL2016597)
Affinity DataIC50:  96nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380432(CHEMBL2018469)
Affinity DataIC50:  152nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380416(CHEMBL2018482)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380440(CHEMBL2018477)
Affinity DataIC50:  181nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380429(CHEMBL2018464)
Affinity DataIC50:  211nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380416(CHEMBL2018482)
Affinity DataIC50:  213nMAssay Description:Inhibition of human CYP2C9 using tolbutamide as substrate by LC/MS/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380411(CHEMBL2018465)
Affinity DataIC50:  221nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380426(CHEMBL2018461)
Affinity DataIC50:  228nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380442(CHEMBL2018479)
Affinity DataIC50:  239nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced cAMP response after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50380414(CHEMBL2018467)
Affinity DataIC50:  284nMAssay Description:Antagonist activity at S1P1 receptor expressed in HEK293 cells assessed as inhibition of S1P-induced tango beta-arrestin recruitment preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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