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Found 111 with Last Name = 'shudo' and Initial = 'k'
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.0400nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076331(1-(hydroxymethyl)-12-(4-hydroxyphenyl)-1,12-dicarb...)
Affinity DataKi:  0.100nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076330(1-(4-hydroxyphenyl)-1,12-dicarba-closo-dodecaboran...)
Affinity DataKi:  0.400nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50076332(1-amino-12-(4-hydroxyphenyl)-1,12-dicarba-closo-do...)
Affinity DataKi:  0.650nMAssay Description:In vitro inhibition of [6,7-3H]-17beta-estradiol binding to human estrogen receptor alphaMore data for this Ligand-Target Pair
Ligand InfoCHEMBLPC sid
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  1nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064090((S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetra...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  3.30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  3.80nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  4.10nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  5.90nMAssay Description:Selective activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  6.5nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  8.30nMAssay Description:Selective activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  11nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073876((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-met...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  12nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064092(5'-hydroxymethyl-2'-isopropyl-1',4,4-trimethyl-(2'...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  16nMAssay Description:Selective activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073875((1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064094(5'-hydroxymethyl-2'-isopropyl-1'-methyl-(2'S,5'S)-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073873((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-d...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  50nMAssay Description:Selective activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  54nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064093((7S,10S)-10-Hydroxymethyl-7-isopropyl-4,4,6-trimet...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290875((S)-13-Hydroxymethyl-10-((S)-isopropyl)-3,9,12-tri...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  120nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  130nMAssay Description:Selective activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  180nMAssay Description:Selective activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073878((4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061616(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  220nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50290877((3S,6S)-6-Hydroxymethyl-3-isopropyl-4-tetradecyl-p...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]-PDBu from Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  330nMAssay Description:Agonisticactivity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  400nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  490nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073872((4S,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073877((4S,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073871((4R,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073870((4R,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  500nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  620nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  640nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor beta(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  680nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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