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Found 180 with Last Name = 'slomczynska' and Initial = 'u'
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074653(CHEMBL385812 | R-K-K-Y-(Ach)-Y-R-R-K-NH2)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM559872(US11375716, Soraphen A)
Affinity DataIC50:  45.8nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074638(CHEMBL443574 | R-K-K-Y-K-Y-R-R-K-NH2)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429101(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  60nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429101(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  60nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074648(CHEMBL268790 | R-K-K-Y-(Ach)-(Ach)-R-R-K-NH2)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase 1(Homo sapiens (Human))
Monsanto Technology

US Patent
LigandPNGBDBM495026(2-(5-(3-chloro-4- phenylquinolin-2- yl)thiophen-2-...)
Affinity DataIC50:  110nMAssay Description: Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429403(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  113nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429403(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  113nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429101(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  116nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429101(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  119nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429101(2-((3-cyano-4-(4- methoxyphenyl)-6-(thiophen- 2-yl...)
Affinity DataIC50:  119nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074635(CHEMBL425624 | R-K-K-Y-K-P-R-R-K-NH2)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM559877(US11375716, Formula Ia-xiv-e1)
Affinity DataIC50:  122nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase 1(Homo sapiens (Human))
Monsanto Technology

US Patent
LigandPNGBDBM495028(2-(5-(4-phenylquinolin-2- yl)thiophen-2-yl)acetic ...)
Affinity DataIC50:  145nMAssay Description: Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074644(CHEMBL409544 | R-K-K-Y-K-F-R-R-K-NH2)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074657(CHEMBL267348 | R-K-K-Y-K-S-R-R-K-NH2)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074642(CHEMBL262895 | R-K-K-Y-K-I-R-R-K-NH2)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074637(CHEMBL265891 | R-K-K-Y-K-M-R-R-K-NH2)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase 1(Homo sapiens (Human))
Monsanto Technology

US Patent
LigandPNGBDBM495021(2-(4-(4-phenylquinolin-2- yl)phenoxy)acetic acid |...)
Affinity DataIC50:  165nMAssay Description: Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429402(2-((3-cyano-4-(4- methoxyphenyl)-6-(1- oxidothioph...)
Affinity DataIC50:  196nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429402(2-((3-cyano-4-(4- methoxyphenyl)-6-(1- oxidothioph...)
Affinity DataIC50:  196nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074639(CHEMBL404932 | R-K-K-Y-K-W-R-R-K-NH2)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429396(2-((4-(4-bromophenyl)-3- cyano-6-(thiophen-2- yl)p...)
Affinity DataIC50:  212nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429396(2-((4-(4-bromophenyl)-3- cyano-6-(thiophen-2- yl)p...)
Affinity DataIC50:  212nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074652(CHEMBL216528 | R-K-K-Y-K-K-R-R-K-NH2)
Affinity DataIC50:  220nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429401(2-((3-cyano-4-(thiophen-2- yl)-5,6,7,8- tetrahydro...)
Affinity DataIC50:  249nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429401(2-((3-cyano-4-(thiophen-2- yl)-5,6,7,8- tetrahydro...)
Affinity DataIC50:  249nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429285(2-((3-cyano-4,6- diphenylpyridin-2-yl)thio)-2- phe...)
Affinity DataIC50:  266nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429285(2-((3-cyano-4,6- diphenylpyridin-2-yl)thio)-2- phe...)
Affinity DataIC50:  266nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074646(CHEMBL415435 | R-K-K-Y-K-(Ach)-R-R-K-NH2)
Affinity DataIC50:  270nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM96465((3-Cyano-4-thiophen-2-yl-5,6,7,8-tetrahydro-quinol...)
Affinity DataIC50:  274nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM96465((3-Cyano-4-thiophen-2-yl-5,6,7,8-tetrahydro-quinol...)
Affinity DataIC50:  274nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074649(CHEMBL262286 | R-K-K-Y-K-N-R-R-K-NH2)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074645(CHEMBL265875 | R-K-K-Y-K-H-R-R-K-NH2)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074655(CHEMBL264533 | R-K-K-Y-K-Q-R-R-K-NH2)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074651(CHEMBL262494 | R-K-K-Y-K-G-R-R-K-NH2)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074636(CHEMBL386668 | R-K-K-Y-K-L-R-R-K-NH2)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429390(2-((3-cyano-6-(furan-2-yl)-4- (4-methoxyphenyl)pyr...)
Affinity DataIC50:  345nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429390(2-((3-cyano-6-(furan-2-yl)-4- (4-methoxyphenyl)pyr...)
Affinity DataIC50:  345nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429392(2-((3-cyano-6-(thiophen-2- yl)-4-(p-tolyl)pyridin-...)
Affinity DataIC50:  353nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429392(2-((3-cyano-6-(thiophen-2- yl)-4-(p-tolyl)pyridin-...)
Affinity DataIC50:  353nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074650(CHEMBL412772 | R-K-K-Y-K-V-R-R-K-NH2)
Affinity DataIC50:  360nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM428892(2-((4-(4-chlorophenyl)-3- cyano-6-(thiophen-2- yl)...)
Affinity DataIC50:  370nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM428892(2-((4-(4-chlorophenyl)-3- cyano-6-(thiophen-2- yl)...)
Affinity DataIC50:  370nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50074643(CHEMBL264293 | R-K-K-Y-K-A-R-R-K-NH2)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity against MLCK (smooth muscle myosin light chain kinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429009(2-((3-cyano-4,6-di(thiophen- 2-yl)pyridin-2-yl)thi...)
Affinity DataIC50:  439nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM559878(US11375716, Formula Ia-xiv-e2)
Affinity DataIC50:  480nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Corn smut fungus)
Monsanto Technology

US Patent
LigandPNGBDBM429014(2-((3-cyano-4-phenyl-6- (thiophen-2-yl)pyridin-2- ...)
Affinity DataIC50:  492nMAssay Description:In order to effectively screen out non-specific modulators of pyruvate kinase and lactate dehydrogenase (the coupled portion of the reaction), a PK/L...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetyl-CoA carboxylase(Zea mays)
Monsanto Technology

US Patent
LigandPNGBDBM429014(2-((3-cyano-4-phenyl-6- (thiophen-2-yl)pyridin-2- ...)
Affinity DataIC50:  492nMAssay Description:Ustilago maydis acetyl CoA carboxylase (ACCase) was cloned, expressed, and purified as described (Weatherly et al, Biochem. J., 2004) and the test co...More data for this Ligand-Target Pair
In DepthDetails US Patent
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