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Found 245 with Last Name = 'sokoloff' and Initial = 'p'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81798(CAS_39860-99-6 | NSC_62867 | Pipotiazine)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81793(CAS_316-81-4 | NSC_92178 | Thioproperazine)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81798(CAS_39860-99-6 | NSC_62867 | Pipotiazine)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50241107(1-(3-(4-(5-chloro-2-oxo-2,3-dihydrobenzo[d]imidazo...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132057(CHEMBL1180430 | CHEMBL126128 | N-{4-[4-(2-Methoxy-...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132040(3-(4-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pi...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50077001(1-Benzyl-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperi...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity of compound towards human Dopamine receptor D4 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM78434(2-chloranyl-10-[3-(4-methylpiperazin-1-yl)propyl]p...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132031(3-(4-Bromo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pipe...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132047(3-(4-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81793(CAS_316-81-4 | NSC_92178 | Thioproperazine)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132059(3-(4-Cyano-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pipe...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132060(3-(3-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81796(CAS_122245 | Iodosulpride | NSC_122245)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132012((E)-3-(4-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50007182(4-Chloro-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132013(CHEMBL341542 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132027(3-(2-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132076(3-Benzo[1,3]dioxol-4-yl-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132019(3-(2-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pi...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132070(CHEMBL338552 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132055(3-Furan-2-yl-N-{4-[4-(2-methoxy-phenyl)-piperazin-...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81796(CAS_122245 | Iodosulpride | NSC_122245)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132039(CHEMBL126280 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132050(CHEMBL126749 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132072(3-(4-Formyl-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132067(CHEMBL129465 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.740nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132053(3-(2-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  0.75nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50025206((6,7-Dihydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  0.910nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  0.920nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132022(Biphenyl-4-carboxylic acid [4-((4aS,10bS)-7-hydrox...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132042(3-Benzo[1,3]dioxol-5-yl-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132078(4-Acetyl-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132024(3-(3-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81793(CAS_316-81-4 | NSC_92178 | Thioproperazine)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81796(CAS_122245 | Iodosulpride | NSC_122245)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132081(3-(2,4-Dichloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1.28nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81796(CAS_122245 | Iodosulpride | NSC_122245)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50241107(1-(3-(4-(5-chloro-2-oxo-2,3-dihydrobenzo[d]imidazo...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132061(3-(3,4-Dichloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1.31nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50131926(CHEMBL127400 | CHEMBL129022 | Isoquinoline-3-carbo...)
Affinity DataKi:  1.48nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM50132038(5-Phenyl-penta-2,4-dienoic acid {4-[4-(2-methoxy-p...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
U. 109

Curated by PDSP Ki Database
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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