Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Tested for its inhibitory activity against HMG-CoA reductase transcription in HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.73E+3nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 3.64E+3nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 5.47E+3nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 7.98E+3nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Upjohn Laboratories
Curated by ChEMBL
Upjohn Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Tested for its inhibitory activity against HMG-CoA reductase transcription in HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+4nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.54E+4nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+4nMAssay Description:In vitro inhibition of Fu5AH acyl coenzyme A:cholesterol acyltransferase.More data for this Ligand-Target Pair