Compile Data Set for Download or QSAR
maximum 50k data
Found 270 with Last Name = 'sridhar' and Initial = 'j'
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133235(CHEMBL132720 | Docosanedioic acid ((S)-5-hydroxyme...)
Affinity DataKi:  0.110nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133238(CHEMBL334853 | Hexadecanedioic acid ((S)-5-hydroxy...)
Affinity DataKi:  0.140nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  0.330nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133238(CHEMBL334853 | Hexadecanedioic acid ((S)-5-hydroxy...)
Affinity DataKi:  0.360nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133235(CHEMBL132720 | Docosanedioic acid ((S)-5-hydroxyme...)
Affinity DataKi:  0.380nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133249(CHEMBL133853 | Dodecanedioic acid [(S)-5-hydroxyme...)
Affinity DataKi:  0.480nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of human Protein kinase C epsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  0.780nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  0.930nMAssay Description:Inhibition of human Protein kinase C alpha with [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133243(CHEMBL132612 | Decanedioic acid ((S)-5-hydroxymeth...)
Affinity DataKi:  1.30nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133249(CHEMBL133853 | Dodecanedioic acid [(S)-5-hydroxyme...)
Affinity DataKi:  1.30nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human PKC beta-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human Protein kinase C gamma with [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133238(CHEMBL334853 | Hexadecanedioic acid ((S)-5-hydroxy...)
Affinity DataKi:  1.80nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133235(CHEMBL132720 | Docosanedioic acid ((S)-5-hydroxyme...)
Affinity DataKi:  2.40nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)
Affinity DataKi:  3.70nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133240(CHEMBL135611 | Decanedioic acid ((2S,5S)-5-hydroxy...)
Affinity DataKi:  4.40nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133249(CHEMBL133853 | Dodecanedioic acid [(S)-5-hydroxyme...)
Affinity DataKi:  5.60nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133243(CHEMBL132612 | Decanedioic acid ((S)-5-hydroxymeth...)
Affinity DataKi:  5.80nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133246(CHEMBL335486 | Hexanedioic acid [(S)-5-hydroxymeth...)
Affinity DataKi:  17nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133240(CHEMBL135611 | Decanedioic acid ((2S,5S)-5-hydroxy...)
Affinity DataKi:  22nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133245(CHEMBL134690 | Octanedioic acid ((1S,6S)-5-hydroxy...)
Affinity DataKi:  31nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant C1b domain of murine Protein kinase C delta in presence of [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133243(CHEMBL132612 | Decanedioic acid ((S)-5-hydroxymeth...)
Affinity DataKi:  38nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133248(CHEMBL134413 | Dodecanedioic acid 4-(2-hydroxymeth...)
Affinity DataKi:  45nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133240(CHEMBL135611 | Decanedioic acid ((2S,5S)-5-hydroxy...)
Affinity DataKi:  57nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133246(CHEMBL335486 | Hexanedioic acid [(S)-5-hydroxymeth...)
Affinity DataKi:  68nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50432670(CHEMBL2347914)
Affinity DataKi:  71nMAssay Description:Irreversible inhibition of CYP1A2 (unknown origin)-mediated demethylation of resorufin methyl ether after 5 mins by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50432670(CHEMBL2347914)
Affinity DataKi:  130nMAssay Description:Irreversible inhibition of CYP1A1 (unknown origin)-mediated deethylation of resorufin ethyl ether after 5 mins by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133251(CHEMBL336963 | Tetradecanedioic acid 4-(2-hydroxym...)
Affinity DataKi:  154nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133248(CHEMBL134413 | Dodecanedioic acid 4-(2-hydroxymeth...)
Affinity DataKi:  169nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133245(CHEMBL134690 | Octanedioic acid ((1S,6S)-5-hydroxy...)
Affinity DataKi:  170nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant murine Protein kinase C delta in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133241(CHEMBL339383 | Octanedioic acid 4-(2-hydroxymethyl...)
Affinity DataKi:  174nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133247(CHEMBL337522 | Decanedioic acid 4-(2-hydroxymethyl...)
Affinity DataKi:  208nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50122946(CHEMBL334195 | Hexanoic acid (5-hydroxymethyl-2-is...)
Affinity DataKi:  225nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133244(CHEMBL134287 | Hexadecanedioic acid 4-(2-hydroxyme...)
Affinity DataKi:  254nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133242(CHEMBL448101 | Hexanedioic acid 4-(2-hydroxymethyl...)
Affinity DataKi:  278nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133250(CHEMBL132525 | Docosanedioic acid 4-(2-hydroxymeth...)
Affinity DataKi:  296nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133237(CHEMBL133777 | Nonanoic acid 4-((2S,4R)-2-hydroxym...)
Affinity DataKi:  296nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133246(CHEMBL335486 | Hexanedioic acid [(S)-5-hydroxymeth...)
Affinity DataKi:  320nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133245(CHEMBL134690 | Octanedioic acid ((1S,6S)-5-hydroxy...)
Affinity DataKi:  558nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133234(CHEMBL132714 | N-(5-Hydroxymethyl-2-isopropyl-1-me...)
Affinity DataKi:  4.47E+3nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Bos taurus (bovine))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50133239(CHEMBL334451 | N-(5-Hydroxymethyl-2-isopropyl-1-me...)
Affinity DataKi:  7.86E+3nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50164693(CHEMBL194721 | N*2*-(3H-Benzoimidazol-5-yl)-N*4*-(...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM7646(CHEMBL102926 | Imidazo[1,2-a]pyridine deriv. 6 | N...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM6619(3-[(9bR)-5-oxo-1H,2H,3H,5H,9bH-benzo[a]pyrrolizin-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of CDK4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50164693(CHEMBL194721 | N*2*-(3H-Benzoimidazol-5-yl)-N*4*-(...)
Affinity DataIC50:  2nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM50378826(CHEMBL1241758)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Georgetown University

Curated by ChEMBL
LigandPNGBDBM6939(4-hydroxy-N-({[3-(4-methoxyphenyl)-4-oxo-2H,4H-ind...)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 270 total ) | Next | Last >>
Jump to: