Affinity DataIC50: 0.0390nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition human full length PI3Kdelta catalytic subunit/p85alpha assessed as formation of PIP3 after 30 mins by europium labeled GRP-based TR-FRET a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition human full length PI3Kdelta catalytic subunit/p85alpha assessed as formation of PIP3 after 30 mins by europium labeled GRP-based TR-FRET a...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human full length PI3K p110delta/p85alpha using phosphatidylinositol 3,4,5-trisphosphate as substrate measured after 30 mins by TR-FRET...More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition human full length PI3Kdelta catalytic subunit/p85alpha assessed as formation of PIP3 after 30 mins by europium labeled GRP-based TR-FRET a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition human full length PI3Kdelta catalytic subunit/p85alpha assessed as formation of PIP3 after 30 mins by europium labeled GRP-based TR-FRET a...More data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of renin in plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human recombinant rennin in buffer assessed as accumulation of angiotensin 1 using human tetradecapeptide by immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Inhibition of renin in bufferMore data for this Ligand-Target Pair