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Found 32 with Last Name = 'stepan' and Initial = 'g'
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataIC50:  19nMAssay Description:Inhibition of HSP90 (unknown origin)More data for this Ligand-Target Pair
TargetHistamine H1 receptor(RAT)
Roche Palo Alto

Curated by ChEMBL
LigandPNGBDBM50162859(2,3-Dihydro-benzo[1,4]dioxine-5-carboxylic acid {1...)
Affinity DataIC50:  100nMAssay Description:Concentration for 50% inhibition towards central histamine H1 receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450019(CHEMBL4174251)
Affinity DataKd:  12nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50218665(SANGLIFEHRIN A)
Affinity DataKd:  3.30nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKd:  17nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50230211(CHEMBL4063126)
Affinity DataKd:  48nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450020(CHEMBL4166066)
Affinity DataKd:  24nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450021(CHEMBL4165935)
Affinity DataKd:  22nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450022(CHEMBL4170426)
Affinity DataKd:  79nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450023(CHEMBL4167017)
Affinity DataKd:  10nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450024(CHEMBL4159110)
Affinity DataKd:  470nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450025(CHEMBL4163568)
Affinity DataKd:  55nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450026(CHEMBL4168950)
Affinity DataKd:  4nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450027(CHEMBL4161025)
Affinity DataKd:  5nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450028(CHEMBL4173004)
Affinity DataKd:  9nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450029(CHEMBL4165103)
Affinity DataKd:  10nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450030(CHEMBL4176386)
Affinity DataKd:  5nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450031(CHEMBL4161280)
Affinity DataKd:  5nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450031(CHEMBL4161280)
Affinity DataKd:  5nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450032(CHEMBL4171881)
Affinity DataKd:  5nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450033(CHEMBL4164700)
Affinity DataKd:  11nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450034(CHEMBL4175329)
Affinity DataKd:  23nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450035(CHEMBL4159376)
Affinity DataKd:  8nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450036(CHEMBL4170010)
Affinity DataKd:  11nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataEC50:  5nMAssay Description:Inhibition of reverse transcriptase Y181C mutant in HIV-1 3B infected in human MT4 cells assessed as inhibition of viral replication after 5 days by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50103642(4-(6-amino-5-bromo-2-(4-cyanophenylamino)pyrimidin...)
Affinity DataEC50:  2nMAssay Description:Inhibition of HIV-1 3B reverse transcriptase K103N mutant infected in human MT4 cells assessed as inhibition of viral replication after 5 days by cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50501284(CHEMBL3944697)
Affinity DataEC50:  347nMAssay Description:Inhibition of HIV-1 3B reverse transcriptase K103N mutant infected in human MT4 cells assessed as inhibition of viral replication after 5 days by cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataEC50:  101nMAssay Description:Inhibition of HIV-1 3B reverse transcriptase K103N mutant infected in human MT4 cells assessed as inhibition of viral replication after 5 days by cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50501284(CHEMBL3944697)
Affinity DataEC50: >500nMAssay Description:Inhibition of reverse transcriptase Y181C mutant in HIV-1 3B infected in human MT4 cells assessed as inhibition of viral replication after 5 days by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450018(CHEMBL4162497)
Affinity DataKd:  140nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Czech Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50103642(4-(6-amino-5-bromo-2-(4-cyanophenylamino)pyrimidin...)
Affinity DataEC50:  12nMAssay Description:Inhibition of reverse transcriptase Y181C mutant in HIV-1 3B infected in human MT4 cells assessed as inhibition of viral replication after 5 days by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50450017(CHEMBL4173859)
Affinity DataKd:  19nMAssay Description:Inhibition of Cy5-labeled cyclosporin A binding to full length recombinant human N-terminal His8-tagged Cyclophilin A (1 to 169 residues) expressed i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed