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Found 1022 with Last Name = 'sugimoto' and Initial = 'k'
TargetAldo-keto reductase family 1 member B10(Homo sapiens (Human))
Gifu Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50442489(CHEMBL2440417)
Affinity DataKi:  1.30nMAssay Description:Competitive inhibition of wild-type human recombinant N-terminal His6-tagged AKR1B10 expressed in Escherichia coli using geraniol as substrate by dou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395732(CHEMBL2164462)
Affinity DataIC50:  0.00200nMAssay Description:Inhibition of human activated TAFI using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395730(CHEMBL2164450)
Affinity DataIC50:  0.0250nMAssay Description:Inhibition of human activated TAFI using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395732(CHEMBL2164462)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of pig pancreatic carboxypeptidase B using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132916(US8846746, 194)
Affinity DataIC50:  0.700nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132862(US8846746, 132)
Affinity DataIC50:  0.900nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133145(US8846746, 463)
Affinity DataIC50:  1.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132882(US8846746, 154)
Affinity DataIC50:  1.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxypeptidase B(Sus scrofa)
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395737(CHEMBL2164457)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of pig pancreatic carboxypeptidase B using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395735(CHEMBL2164459)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human activated TAFI using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132870(US8846746, 140)
Affinity DataIC50:  1.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxypeptidase B(Sus scrofa)
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395735(CHEMBL2164459)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of pig pancreatic carboxypeptidase B using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132856(US8846746, 126)
Affinity DataIC50:  1.20nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132915(US8846746, 193)
Affinity DataIC50:  1.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132874(US8846746, 144)
Affinity DataIC50:  1.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132929(US8846746, 208)
Affinity DataIC50:  1.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132860(US8846746, 130)
Affinity DataIC50:  1.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133143(US8846746, 461)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132857(US8846746, 127)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132936(US8846746, 215)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133146(US8846746, 464)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132848(US8846746, 117)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132924(US8846746, 203)
Affinity DataIC50:  1.40nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132868(US8846746, 138)
Affinity DataIC50:  1.5nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133004(US8846746, 302)
Affinity DataIC50:  1.5nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133055(US8846746, 360)
Affinity DataIC50:  1.5nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132803(US8846746, 70)
Affinity DataIC50:  1.60nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133147(US8846746, 465)
Affinity DataIC50:  1.70nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132809(US8846746, 76)
Affinity DataIC50:  1.70nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132869(US8846746, 139)
Affinity DataIC50:  1.70nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133134(US8846746, 452)
Affinity DataIC50:  1.70nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133135(US8846746, 453)
Affinity DataIC50:  1.70nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132759(US8846746, 25)
Affinity DataIC50:  1.80nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133209(US8846746, 534)
Affinity DataIC50:  1.80nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132823(US8846746, 91)
Affinity DataIC50:  1.80nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132832(US8846746, 100)
Affinity DataIC50:  1.90nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxypeptidase B2(Homo sapiens (Human))
Showa Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50395737(CHEMBL2164457)
Affinity DataIC50:  2nMAssay Description:Inhibition of human activated TAFI using Hip-Arg as substrate incubated for 10 mins prior to substrate addition measured after 30 mins by spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133136(US8846746, 454)
Affinity DataIC50:  2nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132810(US8846746, 77)
Affinity DataIC50:  2nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133116(US8846746, 426)
Affinity DataIC50:  2.05nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133142(US8846746, 460)
Affinity DataIC50:  2.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132944(US8846746, 227)
Affinity DataIC50:  2.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133208(US8846746, 533)
Affinity DataIC50:  2.10nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133200(US8846746, 523)
Affinity DataIC50:  2.15nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133024(US8846746, 324)
Affinity DataIC50:  2.20nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132834(US8846746, 102)
Affinity DataIC50:  2.20nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132935(US8846746, 214)
Affinity DataIC50:  2.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133131(US8846746, 449)
Affinity DataIC50:  2.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM133206(US8846746, 529)
Affinity DataIC50:  2.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
Japan Tobacco

US Patent
LigandPNGBDBM132940(US8846746, 223)
Affinity DataIC50:  2.30nMT: 2°CAssay Description:The stable cell line expressing human SGLT1 was seeded at 5x104 cells/well on BioCoat Poly-D-Lysine 96 well plate with Lid (Becton Dickinson and Comp...More data for this Ligand-Target Pair
In DepthDetails US Patent
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