Affinity DataKi: 0.000660nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.00500nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.00720nMAssay Description:Tested for binding activity against delta1 opioid receptor using [3H]DPDPE ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0150nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0160nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity was measured by the displacement of [3H]- EK in guinea pig brain membrane of opioid receptor kappaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:The compound was evaluated for binding affinity against Opioid receptor delta 1 in guinea pig brain membrane using [3H]- DPDPE as ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Binding affinity was measured by the displacement of [3H]- DAMGO in guinea pig brain membrane of opioid receptor muMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0470nMAssay Description:Tested for binding activity against delta opioid receptor using [3H]naltridole ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0830nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]-DPDPE (delta 1) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:The compound was evaluated for binding affinity against Opioid receptor delta 1 in guinea pig brain membrane using [3H]- DPDPE as ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:The opioid receptor affinity(Ki) was evaluated by competition with [3H]DSLET (delta 2) on guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity was measured by the displacement of [3H]- DAMGO in guinea pig brain membrane of opioid receptor muMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity was measured by the displacement of [3H]- DADLE in guinea pig brain membrane of opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity was measured by the displacement of [3H]- DAMGO in guinea pig brain membrane of Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity was measured by the displacement of [3H]- DAMGO in guinea pig brain membrane of Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity was measured by the displacement of [3H]- DAMGO in guinea pig brain membrane of opioid receptor muMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Tested for binding activity against mu opioid receptor using [3H]DAMGO ligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Tested for binding activity against kappa opioid receptor using [3H]U-69593 ligandMore data for this Ligand-Target Pair