Affinity DataKi: 0.440nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Inhibition of [3H]-pentazocine binding to Sigma opioid receptor type 1More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 0.680nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2 in cell-intact assayMore data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human PDE7A1 expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: <1nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: <1nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PDE7A expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human PDE7A expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human PDE7A1 expressed in insect cells assessed as inhibition of [3H]cAMP to [3H]AMP hydrolysis after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
Kyoto 607-8042
Curated by ChEMBL
Kyoto 607-8042
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of PDE7A (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kirin Brewery
Curated by ChEMBL
Kirin Brewery
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2More data for this Ligand-Target Pair