Affinity DataKi: 21nMAssay Description:Binding affinity to human HSP90-beta by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of FITC-GDA binding to human HSP90-alpha incubated for 2 hrs followed by FITC-GDA addition and measured after 5 hrs by fluorescence polari...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of FITC-GDA binding to human HSP90-alpha incubated for 2 hrs followed by FITC-GDA addition and measured after 5 hrs by fluorescence polari...More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+4nMAssay Description:Binding affinity to human HSP90-beta by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to GRP94 (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
Taiho Pharmaceutical
Curated by ChEMBL
Taiho Pharmaceutical
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to TRAP1 (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to GRP94 (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
Taiho Pharmaceutical
Curated by ChEMBL
Taiho Pharmaceutical
Curated by ChEMBL
Affinity DataKi: >3.00E+5nMAssay Description:Binding affinity to TRAP1 (unknown origin) by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 11.6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 17.8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 18.9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 21.3nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 22.3nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 22.7nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 22.9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 27.8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 28.5nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 28.5nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 28.9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 30.8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 35nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 35.2nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.;
4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and
5,5'...More data for this Ligand-Target Pair