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Found 1267 with Last Name = 'tang' and Initial = 'd'
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430877(CHEMBL2336480)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430878(CHEMBL2336474)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50243007(2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430876(CHEMBL2336473)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548768(CHEMBL4760823)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430887(CHEMBL2336479)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430886(CHEMBL2336476)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548771(CHEMBL4744856)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430885(CHEMBL2336482)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548767(CHEMBL4756164)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548769(CHEMBL4789054)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430884(CHEMBL2336483)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548768(CHEMBL4760823)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430883(CHEMBL2336484)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548769(CHEMBL4789054)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548768(CHEMBL4760823)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548767(CHEMBL4756164)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430882(CHEMBL2336478)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548767(CHEMBL4756164)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548769(CHEMBL4789054)
Affinity DataKi:  263nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430881(CHEMBL2336477)
Affinity DataKi:  277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548771(CHEMBL4744856)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548770(CHEMBL4748774)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548771(CHEMBL4744856)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548789(CHEMBL4777543)
Affinity DataKi:  389nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548772(CHEMBL4791819)
Affinity DataKi:  407nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548795(CHEMBL4762056)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430880(CHEMBL2336481)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)

Curated by ChEMBL
LigandPNGBDBM50430879(CHEMBL2336475)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548778(CHEMBL4763304)
Affinity DataKi:  575nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548772(CHEMBL4791819)
Affinity DataKi:  603nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548761(CHEMBL4762755)
Affinity DataKi:  617nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548780(CHEMBL4758316)
Affinity DataKi:  617nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548759(CHEMBL4796491)
Affinity DataKi:  646nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548759(CHEMBL4796491)
Affinity DataKi:  646nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548769(CHEMBL4789054)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]-NMS from muscarinic M3 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548772(CHEMBL4791819)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548778(CHEMBL4763304)
Affinity DataKi:  891nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548764(CHEMBL4777127)
Affinity DataKi:  912nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548771(CHEMBL4744856)
Affinity DataKi:  977nMAssay Description:Displacement of [3H]-NMS from muscarinic M3 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548778(CHEMBL4763304)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548770(CHEMBL4748774)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548785(CHEMBL4758635)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548766(CHEMBL4747438)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548785(CHEMBL4758635)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548785(CHEMBL4758635)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548760(CHEMBL4778178)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548795(CHEMBL4762056)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50548789(CHEMBL4777543)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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