TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 9.70nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 214nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 257nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 263nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: 277nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 288nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 288nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 302nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 389nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 407nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 417nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Vanderbilt University Institute Of Imaging Science (Vuiis)
Curated by ChEMBL
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 603nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 617nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 617nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 646nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 646nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 776nMAssay Description:Displacement of [3H]-NMS from muscarinic M3 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 776nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 891nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 912nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 977nMAssay Description:Displacement of [3H]-NMS from muscarinic M3 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M1 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.23E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M2 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.23E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Shanghai Jiao Tong University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.38E+3nMAssay Description:Displacement of [3H]-NMS from muscarinic M4 receptor (unknown origin) expressed in CHO-K1 cell membranes assessed as inhibition constant by radioliga...More data for this Ligand-Target Pair